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List of Publication of Professor Rafat M. Mohareb
1- Activated Nitriles In Heterocyclic Synthesis: A Novel Synthesis of
Pyrimidine, Pyridine and Isoxazole Derivatives.
S. M. Fahmy, N. M. Abed, R. M. Mohareb and M. H. Elnagdi;
Synthesis 6, 490 (1982).
2- Activated Nitriles In Heterocyclic Synthesis: A Novel Synthesis of
Tetrazole Derivatives.
S. M. Fahmy and R. M. Mohareb; Synthesis 6, 478 (1983).
3- Activated Nitriles In Heterocyclic Synthesis: Synthesis of Several
New Pyrimidine and Pyridazine Derivatives.
K. U. Sadek, S. M. Fahmy, R. M. Mohareb and M. H. Elnagdi; J.
Chem. Engin. Data 29, 101 (1984).
4- Activated Nitriles In Heterocyclic Synthesis: A Novel Synthesis of
Polyfunctionally Substituted Pyridine Derivatives.
S. M. Fahmy, S. O. Abd Allah and R. M. Mohareb; Synthesis 11,
976 (1984).
5- Activated Nitriles In Heterocyclic Synthesis: A Novel Synthesis of
Pyridine and Pyridazine Derivatives.
S. M. Fahmy and R. M. Mohareb; Synthesis, 1135 (1985).
6- Activated Nitriles In Heterocyclic Synthesis: A Novel Synthesis of
Pyridazine, Pyrimidine, Pyridine and Pyrano[4,3-b]pyridine
Derivatives.
R. M. Mohareb and S. M. Fahmy; Zeitschrift. Fur Naturforschung
40b, 664 (1985).
7- Oxonitrile In Heterocyclic Synthesis: Some New Approaches for
the Synthesis of Pyridazine and Pyrido[2,3-d]pyridazine
Derivatives.
S. M. Fahmy and R. M. Mohareb; Leibigs Ann. Chem., 1492
(1985).
8- Reaction of Malononitrile and Ethyl Cyanoacetate: A Novel
Synthesis of Polyfunctionally Substituted Pyridine Derivatives.
R. M. Mohareb and S. M. Fahmy; Zeitschrift fur Naturforschung
40b, 1537 (1985).
9- Cyanothioacetamide In Heterocyclic Synthesis: A Novel Synthesis
of 2-Pyridothione Derivatives.
S. M. Fahmy and R. M. Mohareb; Tetrahedron, 41 (2), 687 (1986).
10- Cyanothioacetamide In Heterocyclic Synthesis: A New
Approaches for the synthesis of Pyridothione, Pyrane and
Pyridazine Derivatives.
R. M. Mohareb and S. M. Fahmy; Zeitschrift. Fur Naturforschung,
41b, 105 (1986).
11- Dimerized Ethyl Cyanoacetate In Heterocyclic Dye
Synthesis:
New Pyridine Azodye and tetrazole Dyes.
S. M. Fahmy, R. M. Mohareb and F. A. Abd El-Aal; J. Chem.
Tech.
And Biotechnol. 36, 410 (1986).
12- Polyfunctionally Substituted Pyridines from Cyanoacetamide and
Cyanoacetanilide.
R. M. Mohareb, A. Habashi, H. Z. Shams and S. M. Fahmy; Arch.
Die Pharm. (Weinheim) 320, 599 (1987).
13- Reactions With Acetoacetanilide: New Approaches for the
Synthesis of Polyfunctionally Substituted Pyridine Derivatives.
A. Habashi, N. S. Ibrahim, R. M. Mohareb and S. M. Fahmy;
Leibigs
Ann. Der Chemie 1632 (1986).
14- Nitriles In Heterocyclic Synthesis: New Approaches for the
Synthesis of Pyrazoles, Isoxazoles and Pyrimidines.
N. S. Ibrahim, A. A. Hafez and R. M. Mohareb; Heterocycles, 243,
2085 (1986).
15- The chemistry and Synthetic Potentialities of β-Ketoanildes:
Reaction of Ethyl Cyanoacetate with β-Ketoanilides.
A. Habashi, N. S. Ibrahim, S. M. Sherif, H. Z. Shams and R. M.
Mohareb; Heterocycles 24, 2463 (1986).
16- The Synthetic Potentialities of Nitriles In Heterocyclic
Synthesis.
M. H. Elnagdi, S. M. Sherif and R. M. Mohareb; Heterocvycles,
26, 497 (1987).
17- Reaction of Benzoyl Isothiocyanate with Active Methylene
Reagents: A convenient Synthesisd of Pyrazolo[5,4-c]pyrazole, 1,3-
Oxazine, Thiazole and Pyrimidine Derivatives.
R. M. Mohareb, A. Habashi, N. S. Ibrahim and S. M. Sherif;
Synthesis, 3, 228 (1987).
18- α-Haloketoximes In Heterocyclic Synthesis: Polyfunctionally
Substituted Azoles and Azines from Bromoketoximes.
R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif; Arch.
Die Parm. (Weinheim), 320, 776 (1988).
19- Nitriles In Heterocyclic Synthesis: A new Approaches for
The Synthesis of Thiazoles Derivatives.
N. S. Ibrahim, R. M. Mohareb and M. H. elnagdi; J. Fur Prakt.
Chem. 330, 65 (1988).
20- Nitriles In Heterocyclic Synthesis: 1-Cyanoformamide as a
Precursor for a Variety of Heterocyclic Ring Systems.
S. M. Sherif, R. M. Mohareb, G. E. Elgemeie and R. P. Singh;
Heterocycles, 27, 1579 (1988).
21- Nitriles In Heterocyclic Synthesis: New Approaches For the
Synthesis of Some Pyridine Derivatives.
N. S. Ibrahim, R. M. Mohareb and H. Z. Shams; Zeitschrift. Fur
Naturforschung (1988).
22- The Knoevenagel Reaction of Cyanoacetamide with β-
Ketoanilides: Synthesis of Polyfunctionally Substituted pyridine and
Coumarine Derivatives.
R. M. Mohareb and N. S. Ibrahim; J. fur Prak. Chemie, 331, 367
(1989).
23- One Pot Synthesis of Polyfunctionally Substituted 2,3-
Dihydrothiazoles and Thiazolidines.
R. M. Mohareb, S. M. Sherif, A. A. Abdel-Aal, N. I. A. Sayed;
Leibigs Ann. Der Chemie, 1143 (1990).
24− ω-Bromoacetophenone In Heterocyclic Synthesis: A Convenient
One-pot Synthesis and the Chemical Behaviour of 3-
Bromomethylbenzo[d]isoxazole.
R. M. Mohareb, S. M. Sherif, H. Z. Shams and A. M. El-
Torgoman;
Z. Naturforsch., 45b, 1067 (1990).
25- Heterocyclic Synthesis with Isothiocyanates: Synthesis of
Several
New Polyfunctionally Substituted Thiophene, Thiazole and
Thiazolinone Derivatives.
R. M. Mohareb and S. M. Sherif; Arch. Die Pharm.
(Weinheim),
324, 469 (1991).
26- Reactions With 4-Phenyl-3-thiosemicarbazides: A new
Approaches for the Synthesis of Pyrazole, Thiazole, Pyridine and
Pyrido[3,4-b]pyridine Derivatives.
R. M. Mohareb, S. I. Aziz and I El-Sakka; Sulfur Letters, 13
(5) , 299 (1991).
27- A Convenient One-Step Synthesis of Thiophene, Thieno[3,2-
b]pyridazine, Thieno[3,2-b]pyridine and Thiazole Derivatives.
R. M. Mohareb, S. I. Aziz; Sulfur Letters, 13 (5), 229 (1991).
28- y-Bromoacetoacetanilide In Heterocyclic Synthesis: A
Convenient Synthesis of Polyfunctionally Substituted 2,3-
Dihydrothiazole, Pyridine-2-one, 1,2,3-Thiazine, Oxazolo[3,4-
b]pyridine and Pyrazolo[3,4-b]pyridine Derivatives.
R. M. Mohareb, N. I. Abdel-Sayed and S. M. Sherif;
Phosphorous, Sulfur and Silicon, 63, 119 (1991).
29- The Knoevenagel Reaction of Malononitrile with
Acetylacetone:
New Route of Pyrazole, Pyrazolo[2,3-c]pyridine, Benzene,
Pyridazine and Benzo[c]pyridazine Derivatives.
R. M. Mohareb; Arch. Pharm. Res. 14 (4), 379 (1991).
30- Studies With Polyfunctionally Substituted Pyridazines:
Synthesis of new 4-Coumarin-3-yl-pyridazines.
R. M. Mohareb, H. Z. Shams and M. H. Elnagdi; Gazzeta
Chimica Ital., 122, 41(1992).
31- Phenylisothiocyanate In Heterocyclic Synthesis: Novel
Synthesis of Thiazoles, Thieno[2,3-b]pyridine, Thiophene and
Thieno[3,2-c]pyridazine Derivatives.
R. M. Mohareb; Monatschfte fur Chemie, 123, 341 (1992).
32- One-Pot Synthesis of polyfunctionally Substituted Thiophenes,
Thieno[3,4-d]pyridine Derivatives.
R. M. Mohareb; Gazzetta Chemica Ital., 122, 147 (1992).
33- Novel Synthesis of Coumarin-3-yl-1,3-thiazole, 2-(Coumarin-
3-carbonyl)-thieno[2,3-b]pyridine and 2-(Coumarin-3-carbonyl)-
thiophene Derivatives.
R. M. Mohareb, H. Z. Shams and S. I. Aziz; J. Chem. Research
(S), 154 (1992), (M), 1132 (1992).
34- Reactions of Phenyl Isothiocyanate and Sulfur With Dimeric
Adducts: Novel Synthesis of Thiazoles, Thiazolo[4,5-
d]pyrimidine and Thiazolo[4,5-d]pyridine Derivatives.
R. M. Mohareb, H. Z. Shams and Y. M. El-Kholy;
Phosphorous, Sulfur and Silicon, 70, 317 (1992).
35- Heterocyclic Synthese With Isothiocyanates: A Novel
Synthetic Approach to Polyfunctionally Substituted Pyrazoles
and Their Fused Derivatives.
R. M. Mohareb and S. M. Sherif, Sulfur Letters, 15 (1), 91
(1992).
36- The Uses of Ethyl Cyanobromoacetate In Heterocyclic
Synthesis:
Novel Synthesis of Thiophene, Pyrazolo[3,4-d]thiazole and
thieno[2,3-d]pyridazine Derivatives.
R. M. Mohareb, S. El-Kousy and A. M. El-Torgoman; Collect.
Czech. Chem. Commun. 57, 1747 (1992).
37- Novel Synthesis of 4-Bromo-3-oxo-2-phenylhydrazonobutro-
nitrile and 4-Cyano-3-oxo-2-phenylhydrazonobutyronitrile:
Synthesis of Pyridazine, Thiazole, 1,2,4-Triazine and
Pyrido[2,3-e]-1,2,4-triazine Derivatives.
R. M. Mohareb and N. I. A. El-Sayed; Collect. Czech. Chem.
Commun. 57, 1758 (1992).
38- Reactions of Benzoyl Isothiocyanate With Active Methylene
Reagents: A Novel Synthesis of Thiophene, Thiazoline and
Thieno[2,3-d]pyrimidine Derivatives.
R. M. Mohareb, S. I. Aziz, N. I. El-Sayed and H. Z. Shams;
Chin. Chem. Soc., 39, 181 (1992).
39- The Uses of 4-Phenyl-3-Thiosemicarbazide In Heterocyclic
Synthesis.
R. M. Mohareb, H. Z. Shams and Y. M. Elkholy; Phosphorous,
Sulfur and Silicon, 72, 93 (1992).
40- Studies With Alkylheteroaromatic Carbonitrile: Synthesis of
New Mesoionic Pyridazines, Phthalazines and Thienopyridazines.
R. M. Mohareb, A. M. El-Torgoman, S. I. Aziz, S. M. El-Kousy
and M. Riad; Gazzetta Chimica Ital. 122, 503 (1992).
41- Reactions of Benzoylisothiocyanate With Acetoacetanilide:
Synthesis of Pyrrole, Pyridine, Pyrimidine, Pyrazolo[3,4-
d]pyrimidine, Pyrazolo[3,4-d]pyrimidine, Pyrano[4,3-
d]pyrimidine and Pyrido[4,3-d]oxazine Derivatives.
R. M. Mohareb, S. I. Aziz, N. I. A. El-Sayed and F. Z. Elablak;
Collection Czech. Chem. Commun., 58, 947 (1993).
42- Heterocyclic Synthesis With Enamines: Convenient Syntheses
of Polyfunctionally Substituted Pyrazole, Pyridine, Pyrimidine
and Pyrazolo[3,4-d]pyrimidine Derivatives.
R. M. Mohareb, S. M. Sherif and H. F. Zohdi, J. of The Chin.
Chem. Soc., 40, 181 (1993).
43- Heterocyclic Dye Synthesis: Synthesis and Dyeing
Performance of New Polyfunctional Pyridine Azodye.
R. M. Mohareb, S. M. Sherif and H. Z. Shams; A. Dyest. Rep.,
82(5), 37, 52-53 (1993).
44- Heterocyclic Synthesis With Isothiocyanate: An Expecditious
Synthetic Route to Polyfunctionally Substituted Thiophene,
Pyrazole, Oxazole, 2,3-Dihydrothiazole, 2-(Pyrazol-4-
ylideno)thiazole and 5-(thiazol-2-ylideno)-pyrimidine
Derivatives.
S. M. El-Kousy, R. M. Mohareb and S. M. Sherif; J. Chem.
Research (S), 312 (1993), (M), 1981 (1993).
45- Studies With Polyfunctionally Substituted Heteroaromatic: A
New Route to Polyfunctionally Substituted Mercapto-
phthalazines.
M. H. Elnagdi, R. M. Mohareb, F. A. Abdel-Aal and H. A.
Mohamed, Phosphorous, Sulfur & Silicon, 82, 195 (1993).
46- Heterocyclic Synthesis With Isothiocyanate: An Expeditious
Synthetic Route for Polyfunctionally Substituted 3-(Thiazol-2’-
ylidene)pyridines and their Fused Derivatives.
R. M. Mohareb, H. F. Zohdi, S. M. Sherif and W. W.
Wardakhan; Tetrahedron, 50, 5807 (1994).
47- The Reaction Of Active Methylene Reagents With Sulfur and
Phenyl Isothiocyanate: Novel Synthesis of Thiazole,
Thiazolo[4,5-d]pyrimidine and 4,5’-Bithiazolyl Derivatives.
R. M. Mohareb, W. W. Wardakhan and F. Z. El-Ablack; J.
Chem. Research (S), 126 (1994); J. Chem. Research (M), 0747
(1994).
48- The Reaction of 4-Phenyl-3-Thiosemicarbazide with β-
Bifunctional Compounds: Novel Synthesis of Pyridine and
Pyrazole Derivatives.
Y. M. Elkholy and R. M. Mohareb; Phosphorous, Sulfur &
Silicon, 90, 111 (1994).
49- The Reaction of Carbon Disulphide with 2-Aminoprop-1-ene,
1,1,3-tricarbonitrile: One-Pot Synthesis of thiophenes and their
Fused Derivatives.
R. M. Mohareb and S. M. Sherif; J. Chem. Research (S), 484
(1994).
50- Reaction of Carbon Disulphide With Diethyl 3-Amino-2-
Cyano-2-penten-1,5-Dicarboxylate: A Convenient Synthesis of
Polyfunctionally Substituted Thiophenes and Their Fused
Derivatives.
S. M. Sherif, N. I. Abdel-Sayed, S. M. El-Kousy and R. M.
Mohareb; Monatshefte fur Chemie, 126, 601 (1995).
51- Heterocyclic Synthesis With Isothiocyanate and Sulfur: A
Novel Synthesis of Pyrido[2,3-d]thiazole,
thiazolo[4’,5’:2,3]Pyridino[4,5-d]pyridazine and Thiazolo[4,5-
b]isoquinoline Derivatives.
H. Z. Zohdi, R. M. Mohareb and W. W. Wardakhan;
Phosphorous, Sulfur & Silicon, 101, 179 (1995).
52- Heterocyclic Synthesis With Isothiocyanates: A Convenient
Synthesis of Polyfunctionally Substituted 2,3-Dihydrothiazole,
2-(Pyrazol-4’-yl)-Thaizole, 5-(Thiazol-2’-yl)pyrimidine and
Thiazolo-[3,2-a]pyridine Derivatives.
R. M. Mohareb, S. M. Sherif and A. M. Sami; Phosphorous,
Sulfur & Silicon, 101, 57 (1995).
53- Reaction of Carbon Disulphide With Active Methylene
Reagents:
Novel Synthesis of Thiophene, Thieno[2,3-b]thiophene,
Thieno[3,2-c]pyrazole and Thieno[3,2-b]pyridine Derivatives.
R. M. Mohareb, S. M. Sherif, A. Habashi, N. I. Abdel-Sayed
and S. S. Osman; Collect. Czech. Chem. Commun., 60, 1578
(1995).
54- The Uses of Polyfunctionally Substituted Thiophenes In
Heterocyclic Synthesis: Synthesis of Benzo[b]Thiophene,
Thieno[2,3-b]pyridine Derivatives.
R. M. Mohareb, Y. M. Elkholy and N. I. Abdel-Sayed;
Phosphorous, Sulfur & Silicon, 106, 193 (1995).
55- Studies With Polyfunctionally Substituted Heteroaromatics: The
Reactivity of Alkylazoles Towards Electrophilic Reagents.
S. E. Zayed, S. I. Aziz, A. W. Erian, R. M. Mohareb, E. I. Abou
Elmaged, S. A. Metwally and M. H. Elnagdi; Phosphorous, sulfur
And Silicon, 102, 51 (1995).
56- A Convenient Synthesis of Polyfunctionally Substituted
Benzo[b]thiophen-2-yl-pyrimidine, pyrazole, isoxazole and pyridine
derivatives.
S. M. Sherif, R. M. Mohareb, H. Z. Shams and H. M. M.
Gaber; J. Chem. Res. (S), 434, (M) 2658 (1995).
57- The Reaction of 3-Phenyl-5-Aminopyrazole With Carbon
Disulphide: A Novel Synthesis of 3-(3’-phenylpyrazo-5’-yl)-4-
Phenylpyrazol-2-thione, Pyrazolo[3,4-d]thiazole and
Pyrano[2,3-d]thiazole Derivatives.
R. M. Mohareb, H. F. Zohdi and W. W. Wardakhan; Monatsh.
Fur Chem., 126, 1391 (1995).
58- Synthesis of Some New Thiazolines
S. M. Sherif and R. M. Mohareb, 5th, Ibn Siina International
Conference on Pure and Applied Heterocyclic Chemistry, PIP-22
(1995).
59- Studies with Polyfunctionally Substituted Heteroaromatics:
The Reactivity of Alkylazoles Towards Electrophilic Reagents.
S. E. Zayed, S. I. Aziz, A. W. Erian, R. M. Mohareb, E. A. El-
maged and M. H. Elnagdi, Phophorous, Sulfur & Silicon, 51,
102 (1995).
60- β-Enaminonitrilers in Heterocyclic Sytnthesis: A Novel one-
pot Synthesis of Thiophenes and Their Fused Derivatives.
S. M. Sherif, W. W. Wardakhan and R. M. Mohareb; J. of
Chem. Research (S), 356 (1996), (M), 1970 (1996).
61- Convenient Heterocyclization Reactions With Ethyl 2-amino-
4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate: Synthesis of
Thiazole, Isoxazole, Pyrazole, Pyrimidine and Pyridazine
Derivatives.
H. F. Zohdi, W. W. Wardakhan, S. H. Doss and R. M.
Mohareb; J. of Chem. Research, (S), 440 (1996), (M) 2526
(1996)
62- Reaction of 4-Aryl-3-thiosemicarbazides with Carbon
Disulphide: A Facile Convenient Synthesis of 2,3-
Dihydrothiazoles and their Fused Derivatives.
R. M. Mohareb and S. M. Sherif; J. Heteroatom, 77, 8 (1997).
63- The Uses of 4-Aryl-3-thiosemicarbazide In Heterocyclic
Synthesis: Synthesis of Coumarin, Pyrazole, Thiazole and
Thiophene Derivatives.
R. M. Mohareb, S. S. Ghabrial and W. W. Wardakhan,
Phosphorous, Sulfur & Silicon 134, 119 (1998).
64- Studies
With Polyfunctionally Heteroaromatic Compounds: Synthesis of
Some New Polyfunctionally Substituted Pyrido[3,2-c]pyridines
and Pyrido[2,3-c]pyridazines.
S. M. El-Kousy, R. M. Mohareb, M. Raid and M. H. Elnagdi,
Pak. J. Sci. Ind. Res. 41(20, 81-85 (1998).
65- Reaction of 4-Aryl-3-thiosemicarbazide With Phenylisothio-
cyanate: Synthesis of Thiazole, Pyrazole and Pyrimidine
Derivatives.
R. M. Mohareb, W. W. Wardakhan and D. Fleita; J. Chinese
Chemical Society 46, 97 (1999).
66-Synthetic Potentialities of Thiophene In Heterocyclic Synthesis:
A Novel Synthesis of Thieno[2,3-b]pyridine Derivatives.
R. M. Mohareb, H. Z. Shams, Y. M. El-Khooly and R. Azzam
Phosphorous, Sulfur & Silicon 155, 215 (1999).
67-The Reaction of Cyanoacetic acid Hydrazide With Phenyliso-
Thiocyanate.
R. M. Mohareb, S. I. Aziz, N. I. Abdel-Sayed and A. A.
Elbanna
J. of Chemical Research (S), 10 (1999) & (M) 0101, 0128
(1999).
68- Sultamo-Steroid Analogues Part VII: Synthesis of
Epiandrosterons With Potential Activities.
S. H. Doss, R. M. Mohareb, N. A. Lucca and G. A. Elghany,
Arch. Pharmazie 22, 496 (1999).
69- Sudies of The Synthesis of Chiral nonracemic 3,4-disubstituted
Azepanes, a Formal Synthesis of (+) and (-) Balanol Derivatives.
C. Herdeis, R. M. Mohareb, B. R. Neder and T. F.
Schwabenlander; Tetrahedron Asymmetry 10 (23), 4521
(1999).
70- Reaction of Ethyl 2-Diazo-4,5,6,7-Tetrahydrobenzo[b]-
thiophene 3-Carboxylate With Benzoyl Acetonitrile: Synthesis
of Pyrazoles, Pyridazines, Pyrimidines and Their Fused
derivatives.
R. M. Mohareb, M. H. Mohamed and W. W. Wardakhan;
Phosphorous, Sulfur & Silicon, 167 29 (2000).
71-Reaction of 2-Diazo-4,5,6,7-Tetrahydrobenzo[b]thiophene-3-
Carboxylate With 3-Iminobutyronitrile: Synthesis of Thiophene
and Their Fused Derivatives.
R. M. Mohareb and F. M. Manhi; Heteroat. Chem. 11(6), 403
(2000).
72-The Reaction of 2-Amino-3-Cyano-4,5,6,7-Tetrahydrobenzo-
[b]-Thiophene with Diethyl Malonate: Synthesis of Coumarin,
Pyridine and Thiazole Derivatives.
R. M. Mohareb, F. A. El-Omran and J. Ho; Heteroat. Chem.
12(3), 168 (2001).
73- The Reaction of 2-Amino-3-Cyano-4,5,6,7-Tetrahydrobenzo-
[b]thiophene with Ethyl Acetoacetate: Synthesis of Pyridines,
Pyrazoles and Their Fused Derivatives.
R. M. Mohareb and M. H. Mohamed; Heteroat. Chem. 12(6),
518 (2001).
74- One Pot Synthesis OF Thiazolo-2-Hyhrazone, Pydino[2,3-d]-
Pyridazine, Pyrazolo[3,4-d]Pyridazine And Isoxazolo[4,5-
d]Pydrazine Derivatives.
R. M. Mohareb and D. H. Fleita; J. Heteroatom Chem., 13
(3), 258 (2002).
75- Reaction of 3-Cyano-2-amino-4,5,6,7-tetrahydrobenzo[b]-
Thiophene with Dimeric Adducts.
R. M. Mohareb, F. A. El-Omran and J. Ho; Monatash. Fur
Chemie, 133, 1443 (2002).
76- Synthesis and Biological Effects of New Derivatives of
Benzotriazole as Antimicrobial and Antifungal Agents; F. Al-
Omran, R. M. Mohareb and A. A. El-Khair; J. Heterocyclic Chem.,
39, 877 (2002)
.
77- Enantispecific Synthesis of Carbapentostatins
J. Z. Ho, R. M. Mohareb, J. H. Ahn, T. B. Sim and H.
Rapoport; J. Organic Chemistry 68, 109 (2003).
78- An Efficient Procedure for the Preparation of 4-Substituted-5-
aminoimidazoles
M. McLaughlin, R. M. Mohareb and H. Rapoport; J. Organic
Chemistry 68, 50 (2003).
79- Reaction of
2-Diazo-3-cyano-4,5,6,7-Tetrahydrobenzo[b]thiophene With 3-
Iminobutyronitrile: Synthesis of Pyridazines, thiophenes and
their Fused Derivatives.
K. Hilmy, R. M. Mohareb, A. M. El-Torgoman, Y. Sharawy
Phosphorous, Sulfur & Silicon 178(8), 1667 (2003).
80- Synthesis and study of pigment Aggregation response of Some
Melatonin derivatives.
R. M. Mohareb, S. H. doss, G. A. Abdel- Ghany and N. I.
Louca; Pharmazie 58, 9 (2003).
81- Utility of a 2-Aminothiophene-3-carboxamide in the Synthsis
of Thienopyridines and Thienopyrimidines
R. M. Mohareb, S. M. Sherif, H. M. Gaber, S. S. Ghabrial and S.
I. Aziz; Heteroatom Chemistry, 14(5), 459 (2003).
82- An Efficient Procedure for Preparation of (1S,3R)- and
(1S,3S)-1-Amino-3-(hydroxymethyl)cyclopentanes.
H. Rapoport, Y. Ghen, R. M. Mohareb, J. H. Ahn, T. B. Sim
and J. Z. Ho; Chem. Pharm. Bull. 51 (10) 1153-1156 (2003).
83- - Synthesis and Study of Pigment aggregation response of
some melatonin derivatives.
S. H. Doss, R. M. Mohareb, G. A. Elmegeed and N. A. Luoca;
Pharmazie 58, 9 (2003).
84- Heterocyclic Synthesis With Ethyl a-(3-carbamoyl-4,5,6,7-
tetrahydrobenzo[b]thiophen-2-ylhydrazono)acetates: An
Expeditious Synthetic Approach to Polyfunctionally Substituted
Pyran, Pyridine and Pyridazine derivatives.
R. M. Mohareb, S. M. Sherif, H. M. Gaber, S. S. Ghabrial and S.
I. Aziz; Heteroatom Chemistry, 15(4), 300 (2004).
86- Thiophenohydrazonoacetate in Heterocyclic synthesis
R. M. Mohareb, S. M. Sherif, H. M. Gaber, S. S. Ghabrial, S. I.
Aziz; Heteroatom Chem. 15, 15 (2004).
87- Synthesis of Some Novel Heterocyclic Steroids of Potential
Biological Activities: Synthesis of Isoxazolo, Pyrazolo,
Thieno and Phthalazine Derivatives of Epi-Androsterone.
S. H. Doss, R. M. Mohareb and G. A. Elmegeed, Arch.
Pharmazie in press (2004).
88- Uses of 5,5-Dimethyl-7-oxocyclohexeno[b]thiophene
Derivatives in Heterocyclic Synthesis.
D. H. Fleita, A. H. El-Banna and R. M. Mohareb; Phosphorus,
Sulfur& Silicon, 180, 2315 (2005).
89- Acycloaddition Approach to the Curing of ployimides via a
Precursor containing a Thiophene-S,S-dioxide.
A. Maggarosy, R. M. Mohareb and J. Z. Ho; Heteroatom Chem., 17(4),
1, 2006.
90- Synthesis, Structure Elucidation, and Biological Evaluation of
Some Fused and/or Pendant Thiophene, Pyrazole, Imidazole, Thiazole,
Triazole, Triazine, and Coumarin Systems Based on Cyanoacetic 2-
[(Benzoylamino)thioxomethyl] Hydrazide
H. Z. Shams, R. M. Mohareb, M. H. Helal and A. E. Mohamoud;
Phosphoros, Sulfur and Silicon, 182, 237 (2007).
91- Synthesis of thiophenes, azoles and azines with potential biological
activity by employing the versatile heterocyclic precursor N-
benzoycyanoacetylhydrazine
R. M. Mohareb, J. Z. Ho and F. E. Elfarouk; Journal of the Chinese
Chemical Society, 54, 1053, 2007.
92- The reaction of cyanoacetylhydrazine with ω-bromoacetophenone:
Novel Synthesis of 1,3,4-Oxadiazine, Pyridazine and Coumarin
derivatives
R. M. Mohareb, R. A. Ibrahim
and J. Z. Ho; J of the Chilean Chemical
Society, 52(1), 1076 (2007).
93- USESE OF 1-CYANOACETYL-4-PHENYL-3-THIOSEMICARBAZIDE IN
HETEROCYCLIC SYNTHESIS: SYNTHESIS OF THIAZOLE, COUMARIN
AND PYRIDINE DERIVATIVES WITH ANTIMICROBIAL AND
ANTIFUNGAL ACTIVITIES
R. M. Mohareb, J. Z. Ho and A. A Mohamed; Phosphorus, Sulfur and
silicon, 182, 1661, 2007.
94- Uses of progesterone in steroidal heterocyclic derivatives of
potential antimicrobial activity.
R. M. Mohareb, H. Y. Hana; Acta Pharmaceutica, 58, 29-42 (2008).
96- The reaction of β-amino-α,γ-dicyanocrotononitrile with acetophenone:
synthesis of pyridine, pyridazine and thiophene derivatives with
antimicrobial activities.
R. M. Mohareb, K. A. El-Sharkaway and S. M. Sherif, Acta
Pharmaceutica, 58, 429-444 (2008).
97- Synthesis of New disperse azo dyes based on oxopyridine core.
R. M. Mohareb, H. Z. Shams, M. H. Helal and I. M. Samir, Pigment and
Resin Technology, 17, 299-307 (2008).
98- The Reaction of Cyclohexan-1,3-dione with Cyanomethylenes:
Synthesis of Thiophenes and Their Fused Derivatives with Antifungal
Activities
R. M.Mohareb, S. M. Sherif and H. E. Moustafa, Phosphorous, Sulfur &
Silicon, 184, 2078-2096 (2009).
99- The Reaction of Cyanoacetic Acid Hydrazide with 2-Acetylfuran:
Synthesis of Coumarin, Pyridine, Thiophene and Thiazole Derivatives
with Potential Antimicrobial Activities.
R. M. Mohareb, E. E. Elarab, K. A. El-Sharkawy, Scientia Pharmaceutica,
77, 355-366 (2009).
100- SYNTHESIS OF NOVEL TRYPTOPHAN DERIVATIVES OF
POTENTIAL BIOLOGICAL ACTIVITY
R. M. Mohareb, N. A. Louca, G. A. Elmegeed, H. Y. Hanna, J. of Chilean
Chemical Society, 54, 175-179 (2009).
101- The Reaction of Cyanoacetylhydrazine with ω-Bromo(4-
methyl)acetophenone: Synthesis of Heterocyclic Derivatives
with Antitumor Activity.
R. M. Mohareb, A. M. Abdelazeem, Molecules, 15, 3602-3617 (2010).
102- Synthesis of hydrazide-hydrazone derivatives and their evaluation of
antidepressant, sedative and analgesic agents
R. M. Mohareb, K. A. El-Sharkawy, M. M. Hussein and H. M. El-
Sehrawi, J. of Pharmaceutical Science and Research 2(4), 185-196 (2010).
103- Synthesis of Novel Hybrid Steroids with Potential Biological
Activities: Synthesis of C-17-thiazole, isoxazole, pyrazole, thiophene and
phthalazine derivatives of epi-Androsterone.
Rafat M. Mohareb, Senot H. Doss, Gamal A. Elmegeed, Emad F.
Eskander, CURRENT TOPICS IN STEROID RESEARCH, 2010 (in press).
104- Hydrazide-Hydrazones in the Synthesis of 1,3,4-Oxadiazine, 1,2,4-
Triazine and Pyrazole Derivatives with Antitumor Activities
Rafat M. Mohareb, Rehab A. Ibrahim and H.E. Moustafa, The open
Organic Chemistry Journal, 4, 2010 (in press).