10th EurAsian Meeting

on Heterocyclic Chemistry

Milano Marittima – Cervia, Ravenna (Italy)

September, 15th-19th 2019

Embassy & Boston Hotel, Milano Marittima

With the patronage of:

http://www.sciliguria.it/EAMHC2019/sede.htm

EAMHC-2019

Programme

September, 15th September, 16th September, 17th September, 18th September, 19th

Arrival & Registration

9.00-17.00

9.30-11.30

Oral Session 1

PL2IL1OP1 OP2

9.30-11.30

Oral Session 5

PL5IL6OP7 OP8

9.30-11.00

Oral Session 8

IL9 IL10 IL11

9.30-11.10

Oral Session 10

PL7IL13OP13

11.30-11.50

Coffee Break

11.30-11.50

Coffee Break

11.00-11.30

Coffee Break

11.10-11.40

Coffee Break

11.50-12.40

Oral Session 2

IL2OP3

11.50-12.40

Oral Session 6

IL7OP9

11.30-12.20

Oral Session 9

IL12OP12

11.40-12,30

PL8

Closing Ceremony

18.00

Opening Ceremony

18.30-19.20

PL1

20.00

Welcome Party

12.40-14.00

Lunch

12.40-14.00

Lunch

12.20-13.40

Lunch

Lunch

Free Time

Departure

14.00-16.00

Oral Session 3

PL3IL3OP4 OP5

14.00-16.00

Oral Session 7

PL6IL8OP10 OP11

14.30-19.30

Conference Tour

16.00-16.30

Coffee Break

16,00-16.30

Coffee Break

16.30-18.30

Poster Session

16.30-19.00

Oral Session 4

PL4IL4 IL5 OP6 SP

Free Time

Dinner 20.00

Conference Banquet Dinner

Plenary Lectures PL-1 Victor Kartsev, Alexandr Zubenko, Konstantin Krasnov, Athina Geronikaki, Samvel

Sirakanyan Targeted Synthesis of Natural Compounds Analogs. Novel Reactions and Rearrangements

PL-2 Hiriyakkanavar Ila Design and Development of New Efficient and Greener Strategies for Heterocycle Synthesis

PL-3 Richard Taylor, Aimee Clarke, Hon Ho, James Rossi-Ashton, Will Unsworth From Natural Products to Organic Diversity: Dearomatisation and Spirocycle Synthesis

PL-4 Gabriele Cruciani, Jenny Desantis, Laura Goracci Automatic chemical reaction tracking by LC-HRMS

PL-5 Hussein El-Kashef Why Pyrazole?

PL-6 Teresa M. V. D. Pinho e Melo The Chemistry of Nitrosoalkenes, Azoalkenes and 1-Azadienes in the Synthesis of Heterocyclic

Compounds

PL-7 Silvia Schenone, Maurizio Botta Pyrazolo[3,4-d]pyrimidines as protein kinase inhibitors: development of promising

anticancer agents

PL-8 Jiaxi Xu Ring opening and expansion of three-membered heterocycles

Invited Lectures IL-1 M. Merlani, V. Barbakadze, L. Gogilashvili, L. Amiranashvili

Synthetic analogues of natural biopolymer from Boraginaceae family

IL-2 Maria Fesatidou, Athina Geronikaki, Antonios Gavalas, Phaedra Eleftheriou, Marina

Sokovic Design, synthesis and biological evaluation of new dual acting (antimicrobial/anti-

inflammatory) thiazole/thiadiazole derivatives

IL-3 Luca Bernardi Asymmetric organocatalysis: stereoselective approaches to nitrogen heterocycles

IL-4 Babaev E. V., Koval Ya.I., Rybakov V.B. New trends in the chemistry of oxazoles

IL-5 E. Elizbarashvili, N. Ochkhikidze, T. Matitaishvili, A. Pichkhadze, D. Rizhinashvili Synthesis of Macrocyclic Azo-Azomethines. Problems and Solutions

IL-6 Paolo Lupattelli, Teresa Laurita, Lucia Chiummiento, Maria Funicello Stereoselective access to 2,3-diaryl-2,3-dihydrobenzofurans from trans 2,3-diaryloxiranes

IL-7 Asunción Barbero, Carlos Díez-Poza, Alberto Diez-Varga, Laura Fernández-Peña

and Juan Lión The silyl-Prins cyclization: a versatile approach to O- and N-heterocycles

IL-8 Stefano Superchi Biphenyl dioxolanes and azepines as chiroptical probes for the absolute configuration

assignment to chiral molecules

IL-9 Serena Riela Smart Organic/Inorganic Nanocomposites based on Clay Minerals and Heterocycles for

several applications

IL-10 Andrea Basso Photoinduced multicomponent reactions for the generation of nitrogen-containing

heterocycles

IL-11 Maurizio D’Auria Photochemical isomerization of pentaatomic aromatic heterocycles

IL-12 William P. Unsworth Successive Ring Expansion Reactions for the iterative synthesis of macrocycles

IL-13 Matteo Micucci, Alberto Chiarini, Roberta Budriesi Current Status of Heterocycles in Nutraceuticals

Oral Presentations OP-1 Andrea Trabocchi, Elena Lenci, Riccardo Innocenti, Lorenzo Calugi

Diversity-Oriented Synthesis and chemoinformatic analysis of sp3-rich heterocycles

containing the morpholine ring

OP-2 Gabriella Vitali Forconesi, Lisa Moni, Renata Riva Biocatalysis and MCRs: a useful combination for the synthesis of bio-based

polyfunctionalized heterocycles

OP-3 Fatma H. Al-Awadhi, Valerie J. Paul, Hendrik Luesch Discovery and characterization of 3-amino-6-hydroxy-2-piperidone (Ahp)-containing cyclic

depsipeptides: marine-derived elastase inhibitors targeting invasive breast cancer

OP-4 Alessandro Pinna, Luca Banfi, Chiara Lambruschini Multicomponent reactions involved in a new and efficient synthesis of potential organo-

catalysts

OP-5 Sara Meninno, Alessandra Lattanzi Bi- and multifunctional organocatalysts as powerful tools for the asymmetric synthesis of

seven to three membered heterocycles

OP-6 Cecilia Ciccolini, Lucia De Crescentini, Gianfranco Favi, Fabio Mantellini, Giacomo

Mari, Stefania Santeusanio Divergent construction of fused and non-fused N-polyheterocycles via formal [4+2]

Annulation of Indoles with Cyclic Azoalkenes

OP-7 Sigitas Tumkevicius, Jelena Dodonova, Tomas Serevicius, Rokas Skaisgiris, Irina

Fiodorova, Laimis Jagintavicius, Saulius Jursėnas Pyrimidine-Based Donor-Acceptor Emitters: Synthesis and Optical Properties

OP-8 Alice Benzi, Lara Bianchi, Gianluca Giorgi, Massimo Maccagno, Giovanni Petrillo,

Cinzia Tavani Synthesis of poly-functionalized imidazo[1,2-a]pyridines and fluorescent polycycles starting

from the ring-opening of nitrothiophenes

OP-9 Hon E. Ho, Richard J. K. Taylor, William P. Unsworth Merging π-Acid and Pd Catalysis: Dearomatising Spirocyclisation/Cross-Coupling of

Alkyne-tethered Aromatics

OP-10 Jenny Desantis, Laura Goracci, Aurora Valeri, Gabriele Cruciani Design and synthesis of small molecules PROTACs for the targeted degradation of androgen

receptor

OP-11 Samvel N. Sirakanyan, Domenico Spinelli, Athina Geronikaki, Elmira K. Hakobyan,

Anush A. Hovakimyan New biologically active heterocyclic systems based on the pyrano[3,4-c]pyridines

OP-12 Michele Mancinelli, Angela Pagano, Emanuela Marotta, Andrea Mazzanti, Giovanni

Petrillo, Cinzia Tavani Atropisomeric 4,7-Di(naphthalen1-yl)-5,6-dinitro-1H-indoles: Stereodynamic Analysis

OP-13 Nouria A. Al-Awadi, Asaad S. Mohamed, Osama M. Habib Gas-Phase pyrolysis of benzo- and naphthofuran derivatives

Sponsor Presentations SP-1 Dietmar Glindemann

PTFE (“TEFLON”) Sealing Ring for hermetic greaseless Glass Joints

Poster Presentations PP-1 Batenko Nelli, Gaile Anastasija

Synthesis of dichloropyrido[1,2-a]benzimidazol-8,9-dione derivatives and its optical

properties

PP-2 Khadijah M. Al-Zaydi Synthesis of phosphonium ylide derivatives as precursor for anticancer agents

PP-3 L. Amiranashvili, V. Barbakadze, L. Gogilashvili, M. Merlani Chemical content of different species of Boragenaceae family

PP-4 Laura Goracci, Jenny Desantis, Aurora Valeri, Gabriele Cruciani Understanding PROTACs’ metabolism: the next step towards pharmaceutical applications

PP-5 Alya M. Al-Etaibi, Morsy A. El-Apasery Synthesis and Dyeing Performance of some Novel Biologically Active Pyridone Disperse Dyes

on Polyester Fabrics

PP-6 Dario Telese, Carla Boga, Gabriele Micheletti, Joseph Durante Hemiaminals from amino-azaheterocycles and chloral hydrate as synthons for the access to

novel compounds with potential biological activity

PP-7 Ya. I. Koval, A. A. Borovikov, A. V. Schetinin, V. B. Rybakov, E. V. Babaev Cyclization reactions of allyl / propargyl pyridones derivatives, study of their properties

PP-8 Jessica Ceramella, Alexia Barbarossa, Anna Caruso, Domenico Iacopetta, Annaluisa

Mariconda, Carmela Saturnino, Camillo Rosano, Pasquale Longo, Maria Stefania

Sinicropi Diamine derivatives and dithiourea analogues: new multi-target tools against cancer

PP-9 Meaad Saleh Bagazi, Khadijah M. Al- Zaydi, Norah Faihan AlQahtani A Novel Studies of Dienaminone: Synthesis of Heterocyclic Compounds Using Green

Chemistry Methods

PP-10 G. Panzeca, A. Martorana, A. Lauria, F. Mingoia Reactivity, design and synthesis of new aryl-pyrazol-3-one derivatives of biological interest

PP-11 Alessandra Silvani, Stefano Gazzotti, Marco Manenti, Leonardo Lo Presti Allylation of isatin-derived N-Boc-hydrazones followed by Pd-catalyzed carboamination

reaction: an entry to 3-spiro-pyrazolidyl-oxindoles

PP-12 Samvel N. Sirakanyan, Elmira K. Hakobyan, Domenico Spinelli, Athina Geronikaki,

Anush A. Hovakimyan New unique heterocyclic systems: pyrano[4''',3''':4'',5'']pyrido[3'',2'':4',5']thieno(furo)-

[3',2':4,5]pyrimido[2,1-f][1,2,4]triazin-8-ones

PP-13 Ikram Baba Ahmed, Wassila Hadj Slimane, Zahira Kibou, Noureddine Choukchou-

Braham Synthesis of new tetracyclic derivatives of tacrine

PP-14 Noureddine Choukchou-Braham, Nawel Mehiaoui, Zahira Kibou New and Efficient Synthesis of 3-Cyano-2-pyridones Derivatives

PP-15 Noureddine Choukchou-Braham, Djamila Benznine, Zahira Kibou,

Amina Berichi, Redouane Bachir Gold nanoparticules catalysed synthesis of imidazo[1,2-a]pyridine from 2-aminopyridine and

α-haloketone

PP-16 Wassila Hadj Slimane, Ikram Baba Ahmed, Zahira Kibou, Noureddine Choukchou-

Braham Novel multi-component synthesis of amrinone analogues

PP-17 Stefano Superchi, Patrizia Scafato, Giulia Marsico Absolute stereochemistry and synthesis of naturally occurring pyranopyrandiones

PP-18 Deniz Çakmaz, Ergin Keleş, Mohammed Yahya, Anka Utama Putra, Zeynel

Seferoğlu, Ebru Uğur Aktan, Nurgül Seferoğlu A Novel Series Of Indole-Based Colorimetric Chemosensors

PP-19 Angela Pagano, Hon E. Ho, Richard J. K. Taylor, William P. Unsworth Visible-Light-induced Intramolecular Charge Transfer in the Radical Spirocyclisation of

Indole-tethered Ynones

PP-20 Cinzia Tavani, Alice Benzi, Massimo Maccagno, Angela Pagano, Giovanni Petrillo Pyrrole benzannulation as a way to unusual nitroindoles

PP-21 M. Merlani, N. Nadaraia, L. Amiranashvili1, A. Geronikaki, M. Sokovic N-containing 5α-steroids as antimicrobials