cheminform abstract: facile synthesis of isoquinolines by imination and subsequent...

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ChemInform 2011, 42, issue 34 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim Isoquinoline derivatives R 0420 DOI: 10.1002/chin.201134150 Facile Synthesis of Isoquinolines by Imination and Subsequent Palladacycle-Cat- alyzed Iminoannulation of Internal Alkynes. — Mostly mixtures of the isoquino- lines and indenones are obtained from aldehyde substrates with the former as major ones. A facile protocol for the synthesis of indoles via catalytic annulation of ortho- -iodo- and bromoanilines with internal alkynes is developed [cf. (XIX)]. — (YANG, F.; ZHANG, J.; WU*, Y.; Tetrahedron 67 (2011) 16, 2969-2973, http://dx.doi.org/10.1016/j.tet.2011.02.044 ; Dep. Chem., Zhengzhou Univ., Zhengzhou 450052, Henan, Peop. Rep. China; Eng.) — Y. Steudel 34- 150

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Isoquinoline derivativesR 0420 DOI: 10.1002/chin.201134150

Facile Synthesis of Isoquinolines by Imination and Subsequent Palladacycle-Cat-alyzed Iminoannulation of Internal Alkynes. — Mostly mixtures of the isoquino-lines and indenones are obtained from aldehyde substrates with the former as major ones. A facile protocol for the synthesis of indoles via catalytic annulation of ortho--iodo- and bromoanilines with internal alkynes is developed [cf. (XIX)]. — (YANG, F.; ZHANG, J.; WU*, Y.; Tetrahedron 67 (2011) 16, 2969-2973, http://dx.doi.org/10.1016/j.tet.2011.02.044 ; Dep. Chem., Zhengzhou Univ., Zhengzhou 450052, Henan, Peop. Rep. China; Eng.) — Y. Steudel

34- 150

ChemInform 2011, 42, issue 34 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

ChemInform 2011, 42, issue 34 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim