alkaloid - medchemexpress.com · alkaloid alkaloids are a group of naturally occurring chemical...

Alkaloid

Alkaloids are a group of naturally occurring chemical compounds that mostly contain basic nitrogen atoms, produced by a largevariety of organisms including bacteria, fungi, plants, and animals. This group also includes some related compounds with neutraland even weakly acidic properties. Compounds like amino acid peptides, proteins, nucleotides, nucleic acid, amines, and antibioticsare usually not called alkaloids. Alkaloids have a wide range of pharmacological activities including antimalarial, antiasthma,anticancer, cholinomimetic, vasodilatory, antiarrhythmic, analgesic, antibacterial, and antihyperglycemic activities. Many have founduse in traditional or modern medicine, or as starting points for drug discovery. Other alkaloids possess psychotropic and stimulantactivities, and have been used in entheogenic rituals or as recreational drugs. Alkaloids can be toxic too. Although alkaloids act on adiversity of metabolic systems in humans and other animals, they almost uniformly evoke a bitter taste.

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Alkaloid Inhibitors & Modulators

(+)-Bicuculline (d-Bicuculline) Cat. No.: HY-N0219

(+)-Bicuculline is a light-sensitive competitiveantagonist of .GABA-A receptor

Purity: 99.97%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 50 mg, 100 mg, 250 mg

(+)-Magnoflorine (Magnoflorine; α-Magnoflorine; Thalictrine) Cat. No.: HY-N0334

(+)-Magnoflorine (Magnoflorine) is an aporphinealkaloid found in , withAcoruscalamusanti-fungal activity, reduces the formation of C.

’ biofilm. Anti-antidiabetic andalbicansanti-oxidative activity.

Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg

(+)-SparteineCat. No.: HY-W008350

(+)-Sparteine is a natural alkaloid acting as aganglionic blocking agent. (+)-Sparteinecompetitively blocks in thenicotinic ACh receptorneurons.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 100 mg

(+)-ViroallosecurinineCat. No.: HY-N5002

(+)-Viroallosecurinine, isolated from Securinega as a cytotoxic alkaloid, exhibits a MIC ofvirosa

0.48 μg/mL for and .Ps. Aeruginosa Staph. aureusAntibacterial activity.


(-)-Cephaeline dihydrochloride (NSC 32944) Cat. No.: HY-N2260

(-)-Cephaeline dihydrochloride is an enantiomer ofCephaeline dihydrochloride. Cephaelinedihydrochloride is a selective inhibtorCYP2D6with of 121 μM.IC50


(-)-CorynoxidineCat. No.: HY-N7010

(-)-Corynoxidine is an acetylcholinesteraseinhibitor with an value of 89.0 μM, isolatedIC50

from the aerial parts of .Corydalis speciosa(-)-Corynoxidine exhibits antibacterial activitiesagainst Staphylococcus aureus andmethicillin-resistant S.


(-)-Huperzine A (Huperzine A) Cat. No.: HY-17387

(-)-Huperzine A (Huperzine A), an activeLycopodium alkaloid extracted from traditionalChinese herb, is a potent, selective andreversible acetylcholinesterase (AChE) inhibitorand has been widely used in China for thetreatment of Alzheimer's disease (AD).

Purity: >98.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 5 mg, 10 mg

(-)-Isocorypalmine (Tetrahydrocolumbamine; (S)-Tetrahydrocolumbamine) Cat. No.: HY-N0927

(-)-Isocorypalmine, an alkaloid isolated from, possesses antifungalCorydalis chaerophylla

activity.


(-)-SecurinineCat. No.: HY-N2079

(-)-Securinine is plant-derived alkaloid and alsoa antagonist.GABA receptorA

Purity: >98.0%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 25 mg

(-)-Sparteine ((-)-Lupinidine) Cat. No.: HY-W012185

(-)-Sparteine is a natural alkaloid isolated frombeans.

Purity: >98.0%Clinical Data: No Development ReportedSize: 100 mg

2 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]

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https://www.MedChemExpress.com/(-)-Cephaeline_(dihydrochloride).html

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https://www.MedChemExpress.com/_-_-Isocorypalmine.html

https://www.MedChemExpress.com/_-_-Securinine.html

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(-)-Sparteine sulfate pentahydrate ((-)-Lupinidine (sulfate pentahydrate)) Cat. No.: HY-B1304

(-)-Sparteine sulfate pentahydrate ((-)-Lupinidinesulfate pentahydrate) is a class 1a antiarrhythmicagent and a sodium channel blocker. It is analkaloid, can chelate the bivalents calcium andmagnesium.

Purity: >98.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 50 mg

(-)-SalutaridineCat. No.: HY-N2256

(-)-Salutaridine (Salutaridine) is an alkaloidisolated from the stems of Sinomenium

.acutum


(R)-Fangchinoline (Thalrugosine; Thaligine) Cat. No.: HY-N1372

(R)-Fangchinoline (Thalrugosine), a alkaloids fromgenus exhibits antimicrobial andStephaniahypotensive activity.


(S)-NornicotineCat. No.: HY-W040430

(S)-Nornicotine is a metabolite of nicotine.

Purity: >98%Clinical Data:Size: 5 mg

(±)-10-Hydroxycamptothecin ((±)-10-HCPT) Cat. No.: HY-N0275

(±)-10-Hydroxycamptothecin, an indole alkaloidisolated from Camptotheca acuminate, inhibits theactivity of and has a broadtopoisomerase Ispectrum of anticancer activity.

Purity: >98%Clinical Data: No Development ReportedSize: 25 mg, 50 mg, 100 mg

(±)-Huperzine ACat. No.: HY-17388

(±)-Huperzine A, an active Lycopodium alkaloidextracted from traditional Chinese herb, is apotent, selective and reversibleacetylcholinesterase (AChE) inhibitor and has beenwidely used in China for the treatment ofAlzheimer's disease (AD).

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg

1-Deoxynojirimycin (Duvoglustat) Cat. No.: HY-14860

1-Deoxynojirimycin (DNJ, Duvoglustat) is a potentα-glucosidase inhibitor, suppresses postprandialblood glucose, thereby possibly preventingdiabetes mellitus.

Purity: >98.0%Clinical Data: Phase 2Size: 10 mM × 1 mL, 5 mg, 10 mg, 25 mg, 50 mg

10-Deacetyl-7-xylosyl paclitaxel (10-Deacetyl-7-xylosyltaxol;

10-Deacetylpaclitaxel 7-Xyloside; …) Cat. No.: HY-20584

10-Deacetyl-7-xylosyl paclitaxel is a Paclitaxelderivative with improved pharmacological featuresand higher water solubility.


10-MethoxycamptothecinCat. No.: HY-N0446

10-Methoxycamptothecin is a natural bioactivederivative of camptothecin (CPT) isolated from

, and has beenCamptotheca acuminataconfirmed to possess high anti-cancer properties.


12-EpinapellineCat. No.: HY-N2162

12-Epinapelline is a diterpene alkaloid isolatedfrom . 12-EpinapellineAconitum baikalenseexhibits Anti-inflammatory activity and stimulatesthe growth of colonies from fibroblast precursors.



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2-(Methylamino)-1H-purin-6(7H)-one (N2-methylguanine) Cat. No.: HY-101412

2-(Methylamino)-1H-purin-6(7H)-one(N2-Methylguanine) is a modified nucleoside.2-(Methylamino)-1H-purin-6(7H)-one is anendogenous methylated nucleoside found in humanfluids.

Purity: >98.0%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 50 mg, 100 mg

2-Benzoxazolinone (2-Benzoxazolone; 1,3-Benzoxazol-2(3H)-one;

2-Hydroxybenzoxazole) Cat. No.: HY-W015818

2-Benzoxazolinone is an agentanti-leishmanialwith an of 40 μg/mL against . ALC50 L. donovanibuilding block in chemical synthesis.


3-DeoxyaconitineCat. No.: HY-N2164

3-Deoxyaconitine is a diterpenoid alkaloid,isolated from Debx.Aconitum Carmichaeli


3-Hydroxypicolinic acid (Picolinic acid, 3-hydroxy-

(6CI,7CI,8CI); 2-Carboxy-3-hydroxypyridine) Cat. No.: HY-Y0030

3-Hydroxypicolinic acid is a picolinic acidderivative, and belongs to the pyridine family.

Purity: >97.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 1 g

3-Indoleacetic acid (Indole-3-acetic acid; 3-IAA) Cat. No.: HY-18569

3-Indoleacetic acid (Indole-3-acetic acid) is themost common natural plant growth hormone of theauxin class. It can be added to cell culturemedium to induce plant cell elongation anddivision.

Purity: 99.74%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 g

3-Indolepropionic acidCat. No.: HY-W015229

3-Indolepropionic acid is shown to be a powerfulantioxidant and has potential in the treatment forAlzheimer’s disease.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 1 g

3-Methyladenine (3-MA) Cat. No.: HY-19312

3-Methyladenine is a inhibitor.PI3K3-Methyladenine is a widely used inhibitor of

via its inhibitory effect on class IIIautophagyPI3K.

Purity: 99.84%Clinical Data: No Development ReportedSize: 50 mg, 100 mg, 200 mg, 500 mg

3-MethylxanthineCat. No.: HY-50723

3-Methylxanthine, a xanthine derivative, is acyclic guanosine monophosphate inhibitor,(GMP)with an of 920 μM on guinea-pig isolatedIC50

trachealis muscle.


5,6-Dihydro-5-methyluracil (Dihydrothymine) Cat. No.: HY-N6787

5,6-Dihydro-5-methyluracil (Dihydrothymine), anintermediate breakdown product of thymine, comesfrom animal or plants. 5,6-Dihydro-5-methyluracil(Dihydrothymine) can be toxic when present atabnormally high levels.


5-MethyluridineCat. No.: HY-W009444

5-Methyluridine is a is an endogenous methylatednucleoside found in human fluids.



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6-Biopterin (L-Biopterin) Cat. No.: HY-102015

6-Biopterin (L-Biopterin), a pterin derivative, isa cofactor.NO synthase

Purity: 98.02%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg

6-Chloropurine (6-Chloro-9H-purine) Cat. No.: HY-Y0247

6-Chloropurine is a building block in chemicalsynthesis. Intermediate in the preparation of9-alkylpurines and 6-rnercaptopurine. Antitumoractivities.


6-Methoxy DihydrosanguinarineCat. No.: HY-N4228

6-Methoxy Dihydrosanguinarine is an lkaloidisolated from the fruits of M.cordata. 6-MethoxyDihydrosanguinarine shows strong cytotoxicityagainst MCF-7 and SF-268 cell lines with IC50

values of 0.61 μM and 0.54 μM, respectively.


7-EthylcamptothecinCat. No.: HY-N2108

7-Ethylcamptothecin is one of camptothecinanalogues. camptothecin (CPT), a cytotoxicalkaloid isolated from Camptotheca

, is shown to have strong antitumoracuminateactivity against L1210 leukemia and Walker 256carcinosarcoma models.


7-MethylxanthineCat. No.: HY-W017163

7-Methylxanthine, a methyl derivative of xanthine,is one of the purine components in urinarycalculi.


9-MethoxycamptothecinCat. No.: HY-N6011

9-Methoxycamptothecin (MCPT), isolated from, has antitumor activitiesNothapodytes foetida

through inhibition.topoisomerase9-Methoxycamptothecin (MCPT) induces strong G2/Marrest and in cancer.apoptosis


AaptamineCat. No.: HY-N4225

Aaptamine, a spongean alkaloid isolated from a seasponge Aaptos aaptos, is a competitive antagonistof and activates the p21 promoterα-adrenoceptorin a p53-independent manner.


Acetylcholine chloride (Ach; ACh chloride) Cat. No.: HY-B0282

Acetylcholine (chloride) is a common found in the central andneurotransmitter

peripheral nerve system.

Purity: >99.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 1 g, 5 g

AcetylcorynolineCat. No.: HY-N0759

Acetylcorynoline is the major alkaloid componentderived from , and hasCorydalis bungeanaanti-inflammatory properties.


Acetylseneciphylline N-oxideCat. No.: HY-N6848

Acetylseneciphylline N-oxide is a pyrrolizinealkaloid that is seneciphylline in which thehydroxy hydrogen is replaced by an acetyl groupand the tertiary amino function is oxidised to thecorresponding N-oxide.



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https://www.MedChemExpress.com/7-ethylcamptothecin.html

https://www.MedChemExpress.com/7-Methyl-1H-purine-2,6_3H,7H_-dione.html

https://www.MedChemExpress.com/9-methoxycamptothecin.html

https://www.MedChemExpress.com/aaptamine.html

https://www.MedChemExpress.com/Acetylcholine-chloride.html

https://www.MedChemExpress.com/acetylcorynoline.html

https://www.MedChemExpress.com/acetylseneciphylline-n-oxide.html

Acipimox (K-9321) Cat. No.: HY-B0283

Acipimox is a niacin derivative used as ahypolipidemic agent. Target: Acipimox is a niacinderivative used as a hypolipidemic agent.


AcoforestinineCat. No.: HY-N4163

Acoforestinine is a diterpenoid alkaloid isolatedfrom .Aconitum handelianum


Aconine (Jesaconine) Cat. No.: HY-N0277

Aconine inhibits receptor activator of nuclearfactor (NF)-κB ligand (RANKL)-induced NF-κBactivation.

Purity: 99.23%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg

Adenine (6-Aminopurine; Vitamin B4) Cat. No.: HY-B0152

Adenine is a purine derivative and a nucleobasewith a variety of roles in biochemistry.

Purity: 98.76%Clinical Data: LaunchedSize: 10 mM × 1 mL, 1 g, 5 g

Adenine hemisulfate (6-Aminopurine hemisulfate; Vitamin B4 hemisulfate) Cat. No.: HY-B0152B

Adenine hemisulfate (6-Aminopurine hemisulfate) isa purine derivative with a variety of roles inbiochemistry, including cellular respiration, inthe form of both the energy-rich adenosinetriphosphate (ATP) and the cofactors nicotinamideadenine dinucleotide (NAD) and flavin…


Adenine hydrochloride (6-Aminopurine hydrochloride; Vitamin B4 hydrochloride) Cat. No.: HY-B0152A

Adenine hydrochloride (6-Aminopurinehydrochloride) is a purine derivative with avariety of roles in biochemistry, includingcellular respiration, in the form of both theenergy-rich adenosine triphosphate (ATP) and thecofactors nicotinamide adenine dinucleotide…


AICAR phosphate (Acadesine phosphate; AICA Riboside phosphate) Cat. No.: HY-13417A

AICAR phosphate is an activator of AMP-activatedprotein kinase ( ).AMPK

Purity: 99.49%Clinical Data: Phase 3Size: 10 mM × 1 mL, 50 mg, 100 mg, 200 mg, 500 mg

Ajmalicine (Raubasine) Cat. No.: HY-N1919

Ajmalicine (Raubasine) is found in herbs ofCatharanthus roseus, is an antihypertensive drugused in the treatment of high blood pressure,decreases peripheral resistance and bloodpressure.


Ajmaline (Cardiorythmine; (+)-Ajmaline) Cat. No.: HY-B1167

Ajmaline is an alkaloid that is class Iaantiarrhythmic agent.

Purity: 99.31%Clinical Data: LaunchedSize: 10 mM × 1 mL, 50 mg, 100 mg

AkuammilineCat. No.: HY-N2834

Akuammiline, compound 2, is isolated from isolatedfrom the seeds of .Picralima klaineana

Purity: >98%Clinical Data:Size: 1 mg, 5 mg


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Alfuzosin hydrochloride (SL 77499-10) Cat. No.: HY-B0192A

Alfuzosin hydrochloride is an α1 adrenergicreceptor antagonist used to treat benign prostatichyperplasia (BPH).

Purity: >98%Clinical Data: LaunchedSize: 10 mg, 50 mg

AllocryptopineCat. No.: HY-N1933

Allocryptopine, a derivative oftetrahydropalmatine, is extracted from Corydalis

(Thunb.) Pers. Papaveraceae.decumbensAllocryptopine has antiarrhythmic effects andpotently blocks human ether-a-go-go related gene

current.(hERG)


AloperineCat. No.: HY-13516

Aloperine is an alkaloid in sophora plants such as, which has shownSophora alopecuroides L

anti-cancer, anti-inflammatory and anti-virusproperties. Aloperine is widely used to treatpatients with allergic contact dermatitis eczemaand other skin inflammation in China.


Alpha-SolamarineCat. No.: HY-N1917

Alpha-Solamarine is a glycoalkaloid isolated from.Solanum aculeastrum


Ampiroxicam (CP 65703) Cat. No.: HY-17484

Ampiroxicam(CP65703) is a nonselectivecyclooxygenase inhibitor uesd as anti-inflammatorydrug. Target: COX Ampiroxicam is a non-steroidalanti-inflammatory drug. It is a prodrug ofpiroxicam.


Amsacrine hydrochloride (m-AMSA hydrochloride; acridinyl anisidide hydrochloride) Cat. No.: HY-13551A

Amsacrine hydrochloride (mAMSA hydrochloride) isan inhibitor of , and acts as antopoisomerase IIantineoplastic agent which can intercalates intothe DNA of tumor cells.

Purity: >98%Clinical Data: LaunchedSize: 10 mg, 50 mg, 100 mg

Ancitabine hydrochloride (Cyclocytidine hydrochloride;

Cyclo-CMP hydrochloride; Cyclo-C) Cat. No.: HY-N0093

Ancitabine (hydrochloride) is an importantantileukemia drugs.

Purity: 98.59%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 200 mg, 1 g

Anisodamine (6-Hydroxyhyoscyamine) Cat. No.: HY-N0584

Anisodamine (6-Hydroxyhyoscyamine), a belladonnaalkaloid, is a non-subtype-selective muscarinic,and also a nicotinic cholinoceptor antagonist.


Anisodamine hydrobromide (6-Hydroxyhyoscyamine hydrobromide) Cat. No.: HY-N0584A

Anisodamine hydrobromide (6-Hydroxyhyoscyaminehydrobromide), a belladonna alkaloid, is anon-subtype-selective muscarinic, and also anicotinic cholinoceptor antagonist.


ArborineCat. No.: HY-N7004

Arborine, isolated from ,Glycosmis arboreainhibits the peripheral action of acetylcholineand induces a fall in blood pressure.



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Argatroban (MD-805; MCI-9038; Argipidine) Cat. No.: HY-B0375

Argatroban (MD-805) is a direct, selectivethrombin inhibitor.


Aristolochic acid A (Aristolochic acid I; TR 1736) Cat. No.: HY-N0510

Aristolochic acid A (Aristolochic acid I; TR 1736)is the main component of plant extractAristolochic acids, which are found in variousherbal plants of genus Aristolochia and .Asarum


ArmepavineCat. No.: HY-N6857

Armepavine, an active compound from Nelumbo, exerts not only anti-inflammatory effectsnucifera

on human peripheral blood mononuclear cells, butalso immunosuppressive effects on T lymphocytesand on lupus nephritic mice. Armepavine inhibitsTNF-α-induced MAPK and NF-κB signaling cascades.


ATP disodium salt (Disodium adenosine triphosphate; Adenosine

5'-triphosphate disodium salt) Cat. No.: HY-B0345A

ATP disodium salt is a phosphate-group donor forsubstrate activation in metabolic reactions andthe coenzyme for a large number of kinases.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 1 g, 5 g

Atropine (Tropine tropate; DL-Hyoscyamine) Cat. No.: HY-B1205

Atropine (Tropine tropate) is a competitivemuscarinic acetylcholine receptor (mAChR)antagonist with anti-myopia effect.

Purity: 99.55%Clinical Data: LaunchedSize: 10 mM × 1 mL, 100 mg

Atropine sulfate (Sulfatropinol) Cat. No.: HY-B1205A

Atropine sulfate (Sulfatropinol) is abroad-spectrum and competitive muscarinic

antagonist.acetylcholine receptor (mAChR)

Purity: >98%Clinical Data: LaunchedSize: 100 mg

Atropine sulfate monohydrate (Atropine sulfate hydrate) Cat. No.: HY-B0394

Atropine sulfate monohydrate (Atropine sulfatehydrate) is a broad-spectrum and competitivemuscarinic acetylcholine receptor (mAChR)antagonist with anti-myopia effect.


Azaphen (Azafen; Pipofezin hydrochloride; Pipofezine

hydrochloride) Cat. No.: HY-A0022

Pipofezine(Azafen or Azaphen) is a potentinhibitor of the reuptake of serotonin.


BenazeprilCat. No.: HY-B0093

Benazepril, an angiotensin converting enzymeinhibitor, which is a medication used to treathigh blood pressure.

Purity: >98%Clinical Data: LaunchedSize: 1 g, 5 g

Benfotiamine (S-Benzoylthiamine O-monophosphate) Cat. No.: HY-17374

Benfotiamine is a synthetic S-acyl derivative ofthiamine (vitamin B1); an antioxidant dietarysupplement.



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Benzoylaconine (Isaconitine; Pikraconitin) Cat. No.: HY-N0217

Benzoylaconine(Isaconitine; Pikraconitin) is analkaloid in the Chinese traditional medicine RadixAconiti Lateralis Preparata (Fuzi).


Benzoylhypaconine (Benzoylhypacoitine) Cat. No.: HY-N0850

Benzoylhypaconine is a natural product.


Benzoylmesaconine (Mesaconine 14-benzoate) Cat. No.: HY-N0218

Benzoylmesaconine is the most abundant componentof Wutou decoction, which is widely used in Chinabecause of its therapeutic effect on rheumatoidarthritis.

Purity: 98.40%Clinical Data: No Development ReportedSize: 5 mg, 10 mg

BerbamineCat. No.: HY-N0714

Berbamine is a natural compound extracted fromtraditional Chinese medicine Barberry withanti-tumor, immunomodulatory and cardiovasculareffects. Berbamine is a calcium channelblocker.


Berbamine dihydrochlorideCat. No.: HY-N0714A

Berbamine dihydrochloride is an inhibitor of activity with remarkable anti-myelomaNF-κB

efficacy.


BerberineCat. No.: HY-N0716

Berberine is a natural alkaline, reducesapoptosis, with potent anti-oxidative andanti-inflammatory effect.


Berberine chloride (Natural Yellow 18 chloride) Cat. No.: HY-18258

Berberine chloride is an alkaloid isolated fromthe Chinese herbal medicine Huanglian, as an

. Berberine chloride induces reactiveantibioticoxygen species ( ) generation and inhibits ROS DNA

. Antineoplastic properties.topoisomerase


Berberine sulfateCat. No.: HY-N0716B

Berberine sulfate is a natural alkaline, reducesapoptosis, with potent anti-oxidative andanti-inflammatory effect.


Berberrubine chlorideCat. No.: HY-125850

Berberrubine chloride is an active metabolite ofberberine, attenuates ulcerative colitis in micemodel.


Betaine hydrochloride (Betaine chloride) Cat. No.: HY-N0739

Betaine hydrochloride is a natural compound foundin many foods and also an active methyl-donorwhich can maintain normal DNA methylationpatterns.

Purity: >98.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 10 g


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BoldineCat. No.: HY-N6973

Boldine is an aporphine isoquinoline alkaloidextracted from the root of and alsoLitsea cubebapossesses these properties, including antioxidant,anti-inflammatory and cytoprotective effects.


Brevianamide F (Cyclo(L-Pro-L-Trp)) Cat. No.: HY-100385

Brevianamide F , also known ascyclo-(L-Trp-L-Pro), belongs to a class ofnaturally occurring 2,5-diketopiperazines.

Purity: 99.49%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg, 100 mg

Brofaromine (CGP 11305A) Cat. No.: HY-13339

Brofaromine (CGP 11305A) is a monoamine oxidase( ) inhibitor with of 0.2μM forMAO IC50

.MAO-A

Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 20 mg

Bullatine ACat. No.: HY-N5025

Bullatine A (BLA), a diterpenoid alkaloid of the, possesses anti-rheumatic,genus Aconitum

anti-inflammatory and anti-nociceptive effects.


Bulleyaconitine ACat. No.: HY-N0239

Bulleyaconitine A is an analgesic andantiinflammatory drug isolated from Aconitumplants; has several potential targets, includingvoltage-gated Na+ channels.


CalycanthineCat. No.: HY-N5121

Calycanthine, the principal alkaloid of the orderCalycanthaceae, has been isolated from a speciesof the genus , and is a central nervousPsychotriasystem toxin, causing convulsions.


CantharidinCat. No.: HY-N0209

Cantharidin, a natural toxin isolated from beetlesin the families Meloidae and Oedemeridae, has beenreported to be toxic to some pests, including thediamondback moth.

Purity: >98.0%Clinical Data: Phase 2Size: 10 mM × 1 mL, 25 mg, 50 mg, 100 mg, 500 mg

Capsaicin ((E)-Capsaicin) Cat. No.: HY-10448

Capsaicin ((E)-Capsaicin) is a agonist withTRPV1an of 0.29 μM in HEK293 cells.EC50


CarpaineCat. No.: HY-N7016

Carpaine is an alkaloid isolated from Carica papayaLinn with activity,anti-thrombocytopenicexhibits potent activity in sustaining plateletcounts with no acute toxicity. Carpaine has

activity to prevent malaria.anti-plasmodial


CastanospermineCat. No.: HY-N2022

Castanospermine inhibits all forms of α- andβ-glucosidases, especially glucosidase l (requiredfor glucoprotein processing by transfer of mannoseand glucose from asparagine-linked lipids).targetα- and β-glucosidases.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 10 mg, 50 mg, 100 mg


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https://www.MedChemExpress.com/Bulleyaconitine-A.html

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https://www.MedChemExpress.com/Cantharidin.html

https://www.MedChemExpress.com/Capsaicin.html

https://www.MedChemExpress.com/carpaine.html

https://www.MedChemExpress.com/Castanospermine.html

Catharanthine ((+)-3,4-Didehydrocoronaridine) Cat. No.: HY-N0252

Catharanthine is an alkaloid isolated from, inhibitsMadagascar periwinkle

, withvoltage-operated L-type Ca channel2+

anti-cancer and blood pressure-lowering activity.


Catharanthine Tartrate ((+)-3,4-Didehydrocoronaridine Tartrate) Cat. No.: HY-N0252A

Catharanthine Tartrate is an alkaloid isolatedfrom , inhibitsMadagascar periwinkle

, withvoltage-operated L-type Ca channel2+

anti-cancer and blood pressure-lowering activity.


Caulophylline BCat. No.: HY-N6672

Caulophylline B is a fluorenone alkaloid isolatedfrom the roots of Caulophyllum robustumMaxim, affords a low scavenging effect againstDPPH radical.


CefaclorCat. No.: HY-B0198

Cefaclor is an effective antibiotic agent, andspecifically binds to penicillin-binding protein 3( ).PBP 3


Cefsulodin sodiumCat. No.: HY-13588

Cefsulodin sodium salt hydrate is a thirdgeneration β lactam antibiotic and member of thecephems subgroub of antibiotics.


Ceftibuten (Sch 39720) Cat. No.: HY-B0698

Ceftibuten(Sch39720) is a third-generationcephalosporin antibiotic.


Celgosivir (MBI 3253; MDL 28574; MX3253) Cat. No.: HY-16134

Celgosivir (MBI 3253; MDL 28574; MX3253) is an inhibitor; inhibits bovine viralα-glucosidase I

diarrhoea virus (BVDV) with an of 1.27 μM inIC50

assay.in vitro

Purity: >98%Clinical Data: Phase 2Size: 1 mg, 5 mg, 10 mg, 25 mg, 50 mg

CephaelineCat. No.: HY-N4118

Cephaeline is a phenolic alkaloid in Indian Ipecacroots. Cephaeline exhibits potent inhibition ofboth Zika virus (ZIKV) and Ebola virus (EBOV)infections.


Cephalotaxlen ((-)-Cephalotaxine; ZINC19795976) Cat. No.: HY-N0838

Cephalotaxine is an antiviral as well as antitumoragent.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg, 100 mg

CepharanthineCat. No.: HY-N6972

Cepharanthine, an alkaloid derived from Stephania Hayata, with possessescepharantha

anti-inflammatory and antioxidative activities.Cepharanthine attenuates muscle and kidneyinjuries induced by limb ischemia/reperfusion(I/R).



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CetirizineCat. No.: HY-17042

Cetirizine, a second-generation antihistamine, isa major metabolite of hydroxyzine, and a racemicselective H1 receptor inverse agonist used in thetreatment of allergies, hay fever, angioedema, andurticaria.


ChaetocinCat. No.: HY-N2019

Chaetocin is a specific inhibitor of the histonemethyltransferase ( ) SU(VAR)3-9 with an HMT IC50

of 0.6 μM for SU(VAR)3-9. It also inhibitsthioredoxin reductase ( ) with an of 4TrxR IC50

μM.


ChasmanineCat. No.: HY-N1946

Chasmanine is an alkaloid isolated from the rootsof .Aconitum crassicaule


ChelerythrineCat. No.: HY-N2359

Chelerythrine is a natural alkaloid, acts as apotent and selective Ca /phospholopid-dependent2+

antagonist, with an of 0.7 μM.PKC IC50

Chelerythrine has antitumor, antidiabetic andanti-inflammatory activity.


Chelerythrine ChlorideCat. No.: HY-12048

Chelerythrine Chloride is a potent, cell-permeableinhibitor of , with an of 660protein kinase C IC50

nM.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg, 100 mg

ChelidonineCat. No.: HY-N2369

Chelidonine is an isoquinoline alkaloid isolatedfrom , causes G arrestChelidonium majus L. 2/M

and induces caspase-dependent andcaspase-independent , with anticancer andapoptosisantiviral activity.


Chimonanthine ((-)-Chimonanthine) Cat. No.: HY-N5118

Chimonanthine is an alkaloid of Chimonanthus, inhibits tyrosinase and tyrosine-relatedpraecox

protein-1 mRNA expression, amd inhibitsmelanogenesis.


Cinchonidine (α-Quinidine) Cat. No.: HY-N0173

Cinchonidine (α-Quinidine) is a cinchona alkaloidfound in Cinchona officinalis and Gongronemalatifolium. A building block used in asymmetricsynthesis in organic chemistry.


Cinchonine ((8R,9S)-Cinchonine; LA40221) Cat. No.: HY-Y0152

Cinchonine is a natural compound present inCinchona bark. Cinchonine activates endoplasmicreticulum stress-induced apoptosis in human livercancer cells.


CinobufotalinCat. No.: HY-N0880

Cinobufotalin is one of the bufadienolidesprepared from toad venom; has anticancer activity.IC50 value: Target: in vitro: Cinobufotalin(CB)caused significant DNA fragmentation, decrease ofMMP, and an increase in the intracellular Ca(2+)ion and ROS production.



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ColchicineCat. No.: HY-16569

Colchicine is a inhibitor and atubulin disrupting agent. Colchicinemicrotubule

inhibits microtubule polymerization with an IC50

of 3 nM.


Columbamine (Columbamin; Dehydroisocorypalmine) Cat. No.: HY-N0926

Columbamine is a quaternary isoquinoline alkaloidisolated from Argemone mexicana.


Coptisine (Coptisin) Cat. No.: HY-N0430

Coptisine is an alkaloid from Chinese goldthread,and acts as an efficient uncompetitive IDOinhibitor with a value of 5.8 μM and an Ki IC50

value of 6.3 μM.


Coptisine chlorideCat. No.: HY-N0736

Coptisine chloride is an alkaloid from Chinesegoldthread, and acts as an efficient uncompetitive

inhibitor with a value of 5.8 μM and an IDO Ki IC50

value of 6.3 μM.


Coptisine SulfateCat. No.: HY-N0430A

Coptisine Sulfate is an alkaloid from Chinesegoldthread, and acts as an efficient uncompetitive

inhibitor with a value of 5.8 μM and an IDO Ki IC50

value of 6.3 μM.


Cordycepin (3'-Deoxyadenosine) Cat. No.: HY-N0262

Cordycepin, which is a nucleoside derivativeisolated from , inhibits IL-1β-inducedCordyceps

and expression in rheumatoidMMP-1 MMP-3arthritis synovial fibroblasts (RASFs) in adose-dependent manner.


Corydaline ((+)-Corydaline; Corydalin) Cat. No.: HY-N0923

Corydaline is an acetylcholinesterase inhibitorisolated from Corydalis yanhusuo.


CorydineCat. No.: HY-N2571

Corydine is a naturally occurring alkaloid whichcan be extracted from plants such as Croton

leaves. Corydine is efficient onechinocarpusinhibiting (RT) activityreverse transcriptasewith an IC of 356.8 μg/mL.50


CorynolineCat. No.: HY-N0826

Corynoline, isolated from Corydalis incise(Papaveraceae), is a reversible and noncompetitiveacetylcholinesterase ( ) inhibitor with anAChE

of 30.6 μM. Corynoline exhibitsIC50

anti-inflammatory activity by activating .Nrf2


CorynoxeineCat. No.: HY-N0590

Corynoxeine, isolated from the hook of Uncaria, is a potent / inhibitor ofrhynchophylla ERK1 ERK2

key PDGF-BB-induced vascular smooth muscle cells(VSMCs) proliferation.



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https://www.MedChemExpress.com/corynoline.html

https://www.MedChemExpress.com/Corynoxeine.html

CorynoxineCat. No.: HY-N0901

Corynoxine is an enantiomer of Corynoxine B;induces autophagy in different neuronal celllines, including N2a and SHSY-5Y cells.


Corynoxine BCat. No.: HY-N0901A

Corynoxine B is an oxindole alkaloid isolated fromUncaria rhynchophylla (Miq.) Jacks (Gouteng inChinese); a Beclin-1-dependent autophagy inducer.


CorypalmineCat. No.: HY-N0654

Corypalmine is an alkaloid from Corydalis. Corypalmine is an antifungal.chaerophylla


CorytuberineCat. No.: HY-N2570

Corytuberine is an aporphine alkaloid isolatedfrom . CorytuberineDicranostigma leptopodumdisplays cytotoxicity against SMMC-7721 tumorcells.


Cotinine ((-)-Cotinine; (S)-Cotinine; NIH-10498) Cat. No.: HY-B1178

Cotinine is an alkaloid found in tobacco and isalso the predominant metabolite of nicotine, usedas a biomarker for exposure to tobacco smoke.

Purity: 99.42%Clinical Data: Phase 2Size: 10 mM × 1 mL, 50 mg, 100 mg

Crassicauline A (Crassicaulin A) Cat. No.: HY-N1924

Crassicauline A (Crassicaulin A) is a bioactivealkaloid found in roots of Aconitum

. Crassicauline A (Crassicaulin A)carmichaelipossesses feeding deterrent activity against T.

adults with an EC of 1134.5 ppm.castaneum 50


Creatinine (NSC13123) Cat. No.: HY-B0504

Creatinine(NSC13123) is a break-down product ofcreatine phosphate in muscle, and is usuallyproduced at a fairly constant rate by the body.

Purity: >99.0%Clinical Data: Phase 4Size: 10 mM × 1 mL, 1 g, 5 g

CrebanineCat. No.: HY-N2255

Crebanine, an alkaloid from ,Stephania venosainduces G1 arrest and apoptosis in human cancercells. Crebanine exhibits anti-inflammatoryactivity via suppressing MAPKs and Akt signaling.Crebanine also possesses antiarrhythmic effect.


Crotonoside (Isoguanosine) Cat. No.: HY-N0071

Crotonoside is isolated from Chinese medicinalherb, Croton. Crotonoside inhibits andFLT3

, exhibits selective inhibition in acuteHDAC3/6myeloid leukemia (AML) cells. Crotonoside could bea promising new lead compound for the treatment ofAML.


Cyclovirobuxine DCat. No.: HY-N0107

Cyclovirobuxine D (CVB-D) is the main activecomponent of the traditional Chinese medicine Buxus

. Cyclovirobuxine D inducesmicrophylla and attenuates the phosphorylation of autophagy

and .Akt mTOR



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Cytidine (Cytosine β-D-riboside; Cytosine-1-β-D-ribofuranoside) Cat. No.: HY-B0158

Cytidine is a nucleoside molecule that is formedwhen cytosine is attached to a ribose ring,cytidine is a component of RNA.


Cytisinicline (Cytisine; Sophorine; Baptitoxine) Cat. No.: HY-N0175

Cytisinicline (Cytisine) is an alkaloid thatoccurs naturally in several plant genera, such as

and . Cytisinicline (Cytisine)Laburnum Cytisusis a partial agonist of , and partialα4β2 nAChRsto full agonist at β4 containing receptors and α7receptors.


Danofloxacin mesylate (CP 76136-27) Cat. No.: HY-B0501

Danofloxacin mesylate (CP 76136-27) is afluoroquinolone antibacterial for veterinary use.

Purity: 99.59%Clinical Data: LaunchedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg, 100 mg

DauricineCat. No.: HY-N0220

Dauricine, a bisbenzylisoquinoline alkaloid in, possessesAsiatic Moonseed Rhizome

anti-inflammatory activity. Dauricine inhibitscell proliferation and invasion, and inducesapoptosis by suppressing activation in aNF-κBdose- and time-dependent manner in colon cancer.


Daurisoline ((R,R)-Daurisoline) Cat. No.: HY-N0221

Daurisoline is a inhibitor and also anhERG blocker.autophagy


Dehydrocorydaline (13-Methylpalmatine) Cat. No.: HY-N0674

Dehydrocorydaline (13-Methylpalmatine) is analkaloid isolated from traditional Chinese herb

W.T. Wang. DehydrocorydalineCorydalis yanhusuoregulates protein expression of , ;Bax Bcl-2activates , , and inactivatescaspase-7 caspase-8

.PARP

Purity: >98%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg

Dehydrocorydaline chloride (13-Methylpalmatine chloride) Cat. No.: HY-N0674A

Dehydrocorydaline chloride is an alkaloidal thathas anti-inflammatory and anti-cancer activities.Dehydrocorydaline chloride can elevate p38

activation.MAPK


DehydroevodiamineCat. No.: HY-N2106

Dehydroevodiamine is a major bioactive quinazolinealkaloid isolated from , has anEvodiae Fructusantiarrhythmic effect in guinea-pig ventricularmyocytes.


DehydrotomatineCat. No.: HY-N7001

Dehydrotomatine is one of major steroidalglycoalkaloids (SGAs) that accumulate in themature green fruits, leaves and flowers of tomato( ). Dehydrotomatine isSolanum lycopersicumagainst , fungi, insects and animals.bacteria


Delavirdine (U 90152; BHAP-U 90152) Cat. No.: HY-10571

Delavirdine(U 90152) is a potent non-nucleosidereverse transcriptase inhibitor (NNRTI).

Purity: >98%Clinical Data: LaunchedSize: 10 mg, 50 mg, 100 mg, 200 mg


https://www.MedChemExpress.com/Cytidine.html

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https://www.MedChemExpress.com/dehydroevodiamine.html

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https://www.MedChemExpress.com/delavirdine.html

DelsolineCat. No.: HY-N0789

Delsoline, a major alkaloid of Delphinium, has both a curare-likeanthriscifolium Hance

effect and a ganglion-blocking effect and is usedto relieve muscle tension or hyperkinesia. D.


DeltalineCat. No.: HY-N0329

Deltaline is a diterpenoid alkaloid and isolatedfrom plants of the genus Delphinium delavayiFranch.


DendrobineCat. No.: HY-N0638

Dendrobine is an alkaloid isolated from. Dendrobine possessesDendrobium nobile

antiviral activity against , withinfluenza A virusess of 3.39 μM, 2.16 μM and 5.32 μM forIC50

A/FM-1/1/47 (H1N1), A/Puerto Rico/8/34 H274Y(H1N1) and A/Aichi/2/68 (H3N2), respectively.


DenudatineCat. No.: HY-N1982

Denudatine, is primarily isolated from plants ofthe genera Aconitum and Delphinium. Denudatine haseffects on action potential of ventricular fibersand inhibits arrhythmogenic action of aconitine.


Desmethylglycitein (4',6,7-Trihydroxyisoflavone) Cat. No.: HY-N5072

Desmethylglycitein (4',6,7-Trihydroxyisoflavone),a metabolite of daidzein, sourced from Glycine

with antioxidant, and anti-cancermaxactivities.


DetomidineCat. No.: HY-B0163

Detomidine produce dose-dependent sedative andanalgesic effects, is a nonnarcotic, syntheticα2-adrenergic agonist.


DicentrineCat. No.: HY-N6969

Dicentrine is a natural product isolated from theplant with antihypertensiveLindera megaphyllaeffect. Dicentrine is an α -adrenoceptor1

antagonist which has effective against humanhyperplastic prostates.


Dictamine (Dictamnine; Dectamine) Cat. No.: HY-N0849

Dictamnine (Dictamine) has the ability to exertcytotoxicity in human cervix, colon, and oralcarcinoma cells; A natural plant product has beenreported to have antimicrobial activity againstbacteria and fungi.


Dihydralazine sulfateCat. No.: HY-N7065

Dihydralazine sulfate is an antihypertensiveagent.


DihydrocapsaicinCat. No.: HY-N0361

Dihydrocapsaicin is a natural capsaicin, acts as aselective agonist, and also increases p-AktTRPV1levels. Dihydrocapsaicin enhances thehypothermia-induced neuroprotection.



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https://www.MedChemExpress.com/dihydralazine-sulfate.html

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Dihydrochelerythrine (12,13-Dihydrochelerythrine) Cat. No.: HY-N0903

Dihydrochelerythrine is a natural compoundisolated from the leaves of Macleaya microcarpa;has antifungal activity. IC50 value: Target: invitro: Dihydrochelerythrine showed the highestantifungal activity against B.


DihydrolycorineCat. No.: HY-N2403

Dihydrolycorine is isolated from Lycoris radiateHerb with antihypertensive and neuroprotectiveactivities.


DihydropalmatineCat. No.: HY-N4240

Dihydropalmatine is a alkaloid isolated from.Berberis aristata


Dihydrosanguinarine (13,14-Dihydrosanguinarine) Cat. No.: HY-N0902

Dihydrosanguinarine is a natural compound isolatedfrom the leaves of Macleaya microcarpa; hasantifungal and anticancer activity.


Dobutamine hydrochlorideCat. No.: HY-15746

Dobutamine hydrochloride is a sympathomimetic drugused in the treatment of heart failure andcardiogenic shock. Its primary mechanism is directstimulation of β1 receptors of the sympatheticnervous system.


Doxazosin (UK 33274) Cat. No.: HY-B0098

Doxazosin(UK 33274) is a quinazoline-derivativethat selectively antagonizes postsynapticα1-adrenergic receptors.


Ecteinascidin 770 (Ecteinascidine 770; Et-770) Cat. No.: HY-101191

Ecteinascidin 770 (ET-770) is a1,2,3,4-tetrahydroisoquinoline alkaloid withpotent anti-cancer activities; inhibits U373MGcells with an of 4.83 nM.IC50

Purity: 98.82%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 1 mg

Efavirenz (DMP 266; EFV; L-743726) Cat. No.: HY-10572

Efavirenz is a potent inhibitor of the wild-type with a of 2.93 nM andHIV-1 reverse transcriptase Ki

exhibits an of 1.5 nM for the inhibition ofIC95

HIV-1 replicative spread in cell culture.

Purity: 99.99%Clinical Data: LaunchedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg

Ellipticine (NSC 71795) Cat. No.: HY-15753

Ellipticine (NSC 71795) is a potent antineoplasticagent; inhibits activities.DNA topoisomerase II

Purity: >98%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 50 mg, 100 mg

Ellipticine hydrochloride (NSC 71795 (hydrochloride)) Cat. No.: HY-15753A

Ellipticine (NSC 71795) hydrochloride is a potentantineoplastic agent; inhibits DNA topoisomerase

activities.II



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https://www.MedChemExpress.com/Ellipticine.html

https://www.MedChemExpress.com/Ellipticine-hydrochloride.html

Emetine dihydrochlorideCat. No.: HY-B1479A

Emetine (dihydrochloride) is an anti-protozoaldrug previously used for intestinal and tissueamoebiasis.


Enniatin BCat. No.: HY-N3806

Enniatin B is a mycotoxin. Enniatin BFusariuminhibits acyl-CoA: cholesterol acyltransferase( ) activity with an of 113 μM in anACAT IC50

enzyme assay using rat liver microsomes. EnniatinsB decreases the activation of (p44/p42).ERK


Enniatin B1Cat. No.: HY-N3807

Enniatin B1 is a mycotoxin. EnniatinFusariumB1 inhibits acyl-CoA: cholesterol acyltransferase( ) activity with an of 73 μM in anACAT IC50

enzyme assay using rat liver microsomes. EnniatinB1 crosss the blood-brain barrier.


EpiberberineCat. No.: HY-N0226

Epiberberine is an alkaloid isolated from Coptis, acts as a potent and chinensis AChE BChE

inhibitor, and a non-competitive inhibitor,BACE1with s of 1.07, 6.03 and 8.55 μM,IC50

respectively.


Epiberberine chlorideCat. No.: HY-N0226A

Epiberberine chloride is an alkaloid isolated from, acts as a potent and Coptis chinensis AChE BChE

inhibitor, and a non-competitive inhibitor,BACE1with s of 1.07, 6.03 and 8.55 μM,IC50

respectively.


Etimizol (Ethimizole; Ethymisol; Ethymisole) Cat. No.: HY-13918

Etimizol(Ethymisole; Antiffine; Ethylnorantifein)was shown to relieve amnesia effectively in theorigin of which there is the hypoxic component(hypobaric hypoxia, actinomycin D, mechanicalinjury of the brain).


Evodiamine ((+)-Evodiamine; d-Evodiamine) Cat. No.: HY-N0114

Evodiamine is an alkaloid isolated from the fruitof Bentham with diverse biologicalEvodia rutaecarpaactivities including anti-inflammatory,anti-obesity, and antitumor.


Fenspiride HydrochlorideCat. No.: HY-A0027

Fenspiride Hcl is an α adrenergic and H1 histaminereceptor antagonist.


Flaconitine (Acetylaconitine; 3-Acetylaconitine) Cat. No.: HY-N0276

Flaconitine is isolated from the ammoniumhydroxide wetted root of Gay.A.szechenyianumFlaconitine is considered to be a NF-κBinhibitor.


Flupirtine (D 9998) Cat. No.: HY-17001A

Flupirtine(D 9998) is a selective neuronalpotassium channel opener that also has NMDAreceptor antagonist properties.



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https://www.MedChemExpress.com/Fenspiride-Hydrochloride.html

https://www.MedChemExpress.com/Flaconitine.html

https://www.MedChemExpress.com/flupirtine.html

Fluvoxamine (DU-23000) Cat. No.: HY-B0103

Fluvoxamine (DU-23000) is an antidepressant whichfunctions pharmacologically as a selectiveserotonin reuptake inhibitor.


Foresaconitine (Vilmorrianine C) Cat. No.: HY-N0851

Foresaconitine(Vilmorrianine C) is anorditerpenoid alkaloid isolated from theprocessed tubers of Aconitum carmichaeli.

Purity: >98.0%Clinical Data: No Development ReportedSize: 5 mg, 10 mg

Fosinopril sodium (SQ28555) Cat. No.: HY-B0382

Fosinopril Sodium is the ester prodrug of anangiotensin-converting enzyme (ACE) inhibitor,used for the treatment of hypertension and sometypes of chronic heart failure.


Fumitremorgin C (12α-Fumitremorgin C) Cat. No.: HY-N2143

Fumitremorgin C is a potent and selective inhibitor.ABCG2/BRCP

Purity: 99.63%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 250 μg, 1 mg

Galanthamine (Galantamine) Cat. No.: HY-76299

Galanthamine is a potent acetylcholinesterase( ) inhibitor with an of 500 nM.AChE IC50


Galanthamine hydrobromide (Galantamine hydrobromide) Cat. No.: HY-A0009

Galanthamine hydrobromide is a long-acting,centrally active acetylcholinesterase(AChE)inhibitor (IC50 = 410 nM) and allostericpotentiator at neuronal nicotinic ACh receptors.


Gatifloxacin hydrochloride (AM 1155 hydrochloride; BMS

206584-01 hydrochloride; PD 135432 hydrochloride) Cat. No.: HY-10581A

Gatifloxacin (hydrochloride) is an antibiotic ofthe fourth-generation fluoroquinolone family, itinhibits the bacterial enzymes DNA gyrase andtopoisomerase IV.


Geissoschizine methyl etherCat. No.: HY-N2411

Geissoschizine methyl ether, a major indolealkaloid found in hook, is a major activeUncariacomponent of Yokukansan with psychotropic effects.Geissoschizine methyl ether is potent 5-HT1A

agonist.receptor


GelsemineCat. No.: HY-N0388

Gelsemine, an alkaloid from the Chinese herb, is effective in mitigatingGelsemium elegans

chronic pain. Antinociceptive and hypnoticeffects.


Glycoursodeoxycholic acid (Ursodeoxycholylglycine) Cat. No.: HY-N1424

Glycoursodeoxycholic acid, a acyl glycine and abile acid-glycine conjugate, is a metabolite ofursodeoxycholic acid.



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Gramine (Donaxine) Cat. No.: HY-N0166

Gramine (Donaxine) is a natural alkaloid isolatedfrom giant reed, acts as an active adiponectin

agonist, with s of 3.2 andreceptor (AdipoR) IC50

4.2 µM for AdipoR2 and AdipoR1, respectively.Gramine is also a human and mouse β2-Adrenergic

agonist.receptor (β2-AR)


Granisetron (BRL 43694) Cat. No.: HY-B0071

Granisetron (BRL 43694) is a serotonin 5-HT3receptor antagonist used as an antiemetic to treatnausea and vomiting following chemotherapy.


Guvacine hydrochlorideCat. No.: HY-100809

Guvacine hydrochloride is an alkaloid from the nutof , acts as an inhibitor of Areca catechu GABA

, and dispalys modest selectivity fortransportercloned GABA transporters with s of 14 μMIC50

(human GAT-1), 39 μM (rat GAT-1), 58 μM (ratGAT-2), 119 μM (human GAT-3), 378 μM (rat…


Halofuginone (RU-19110) Cat. No.: HY-N1584

Halofuginone (RU-19110) is a less-toxic form ofFebrifugine, which is isolated from the plant

. Halofuginone inhibits Dichroa febrifuga prolyl-tRNA in an ATP-dependent manner with a synthetase Ki

of 18.3 nM. Halofuginone attenuates osteoarthritis(OA) by inhibition of activity.TGF-β

Purity: 98.32%Clinical Data: Phase 2Size: 10 mM × 1 mL, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg

Halofuginone hydrobromide (RU-19110 (hydrobromide)) Cat. No.: HY-N1584A

Halofuginone hydrobromide (RU-19110 hydrobromide)is a less-toxic form of Febrifugine, which isisolated from the plant .Dichroa febrifugaHalofuginone inhibits in anprolyl-tRNA synthetaseATP-dependent manner with a of 18.3 nM.Ki


Harmine (Telepathine) Cat. No.: HY-N0737A

Harmine is a natural dual-specificity tyrosinephosphorylation-regulated kinase ( )(DYRK)inhibitor with anticancer and anti-inflammatoryactivities.


HarringtonineCat. No.: HY-N0862

Harringtonine is a natural alkaloidCephalotaxusthat inhibits .protein synthesis

Purity: 99.91%Clinical Data: Phase 3Size: 10 mM × 1 mL, 5 mg, 10 mg

HirsuteineCat. No.: HY-N2197

Hirsuteine is an indole alkaloid extracted from. Hirsuteine non-competitivelyUncaria genus

antagonizes nicotine-mediated dopamine release byblocking ion permeation through nicotinic receptorchannel complexes.


HirsutineCat. No.: HY-N2193

Hirsutine, an indole alkaloid of Uncaria, exhibits anti-cancer activity.rhynchophylla

Hirsutine induces apoptosis and is a potent Denguevirus inhibitor exhibiting low cytotoxicity.


Homoharringtonine (Omacetaxine mepesuccinate; HHT) Cat. No.: HY-14944

Homoharringtonine (Omacetaxine mepesuccinate;HHT)is a cytotoxic alkaloid with antitumor propertieswhich acts by inhibiting .translation elongation



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Hydrastine ((-)-β-Hydrastine; (1R,9S)-β-Hydrastine) Cat. No.: HY-B0927

Hydrastine is a natural alkaloid which is presentin Hydrastis canadensis and other plants of theranunculaceae family.


HydroprotopineCat. No.: HY-N2483

Hydroprotopine is a alkaloid from Hypecoum. Leptopidine can suppress growthleptocarpumand

and induce cytotoxicity in breast cancer cells andthat the cytotoxicity of leptopidine may berelated to its inhibitory effect on fatty acidsynthase expression.


Hydroxy-β-sanshoolCat. No.: HY-N6824

Hydroxy-β-sanshool is an alkylamide exists inZanthoxylum bungeanum oil and Zanthoxylumschinifolium oil.


Hydroxy-γ-sanshoolCat. No.: HY-N6823

Hydroxy-γ-sanshool is an alkylamide exists inZanthoxylum bungeanum oil and Zanthoxylumschinifolium oil.


Hydroxy-α-sanshoolCat. No.: HY-N6825

Hydroxy-α-sanshool is an alkylamide isolatedfrom , acts as a covalent and pepper TRPA1 TRPV1non-covalent agonist, with s of 69 and 1.1EC50

µM, respectively.


HypaconitineCat. No.: HY-N0267

Hypaconitine, an active and highly toxicconstituent derived from Aconitum species, iswidely used to treat rheumatism.


Hypoxanthine (Purin-6-ol; Sarcine) Cat. No.: HY-N0091

Hypoxanthine, a purine derivative, is a potentialfree radical generator and could be used as anindicator of hypoxia.


Indaconitine (15-Deoxyaconitine) Cat. No.: HY-N0788

Indaconitine is a natural product.


Indirubin (Couroupitine B; Indigo red; Indigopurpurin) Cat. No.: HY-N0117

Indirubin (Couroupitine B) is a purple 3,2-bisindole and a stable isomer of indigo isolatedfrom Indigo naturalis (Apiaceae);anti-inflammatory and anticancer activities.

Purity: >98.0%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 250 mg

Indole-3-butyric acid (3-indolebutyric acid) Cat. No.: HY-N0186

Indole-3-butyric acid (3-indolebutyric acid; IBA)is a plant growth auxin and a good rooting agent.It can promote herbs and woody ornamental plantrooting and used for improving fruit rate.

Purity: 99.66%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 5 g, 10 g


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Indole-3-carbinol (I3C; 3-Indolemethanol) Cat. No.: HY-N0170

Indole-3-carbinol (I3C) inhibits activityNF-κBand also is an ( )Aryl hydrocarbon receptor AhRagonist, and an inhibitor of (WWWWP1domain-containing ubiquitin E3 ligase 1).

Purity: >98.0%Clinical Data: Phase 2Size: 10 mM × 1 mL, 200 mg, 1 g

Isatin (Indoline-2,3-dione) Cat. No.: HY-Y0265

Isatin (Indoline-2,3-dione) is a potent inhibitorof with an of 3monoamine oxidase (MAO) IC50

μM. Also binds to central benzodiazepine receptors(IC against clonazepam, 123 μM).50


Isocorynoxeine (7-Isocorynoxeine) Cat. No.: HY-N0775

Isocorynoxeine, an isorhynchophylline-relatedalkaloid, exhibits a dose-dependent inhibition of

receptor-mediated current response with5-HT2A

an of 72.4 μM.IC50


IsorhynchophyllineCat. No.: HY-N0766

Isorhynchophylline (IRN), an alkaloid isolatedfrom Uncaria rhynchophylla, possesses the effectsof lowered blood pressure, vasodilatation andprotection against ischemia-induced neuronaldamage.


Isovaleramide (3-Methylbutanamide) Cat. No.: HY-B1229

Isovaleramide is an active principle on centralnervous system from Valeriana pavonii, as ananticonvulsant. Target in vitro: Isovaleramide(300 μM) exhibits a 42% of inhibition of thebinding of 3H-FNZ to its sites. in vivo:Isovaleramide at 100 mg/Kg, p.

Purity: >98%Clinical Data: No Development ReportedSize: 100 mg

Jervine (11-Ketocyclopamine) Cat. No.: HY-N0836

Jervine(11-Ketocyclopamine) is a naturallyoccuring steroidal alkaloid that causes cyclopiaby blocking sonic hedgehog(Shh) signaling; Jervineis an inhibitor of Smo. IC50 value: Target: sonichedgehog is derived from the Veratrum plantspecies.

Purity: 99.03%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 50 mg

KaracolineCat. No.: HY-N6812

Karacoline, a diterpene alkaloid found in theplant , reduces degradationAconitum kusnezoffiiof the extracellular matrix (ECM) inintervertebral disc degeneration (IDD) via theNF-κB signaling pathway.


Ketanserin tartrate (R41468 tartrate) Cat. No.: HY-10562A

Ketanserin tartrate is a selective 5-HT receptorantagonist. Ketanserin tartrate also blocks hERGcurrent ( ) in a concentration-dependentIhERG

manner ( =0.11 μM).IC50


Kinetin (6-Furfuryladenine; N6-Furfuryladenine) Cat. No.: HY-N0160

Kinetin (N6-furfuryladenine) belongs to a group ofplant growth hormones involved in cell division,differentiation and other physiological processes.

Purity: 99.72%Clinical Data: Phase 4Size: 10 mM × 1 mL, 1 g, 5 g

KoumineCat. No.: HY-N1440

Koumine is an alkaloid separated from Gelsemium, shows potent anti-tumor activity. Koumineelegans

up-regulates the Bax/Bcl-2 ratio and caspase-3expression in human breast cancer cells.



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Kukoamine ACat. No.: HY-N2392

Kukoamine A is a natural occurring sperminederivative, acts as a potent inhibitor of

( , 1.8 μM), withtrypanothione reductase Ki

antihypertensive activity.


Kukoamine BCat. No.: HY-N2393

Kukoamine B is a component of Lycii Cortex, withanti-oxidant, anti-acute inflammatory andanti-diabetic properties.


L-(+)-Abrine (L-Abrine; L-N-Methyltryptophan; N-α-Methyl-L-tryptophan) Cat. No.: HY-N1436

L-(+)-Abrine, a lethal albumin found in Abrus seeds, is an acute toxic alkaloid andprecatorius

chemical marker for abrin.


L-DOPA (Levodopa; 3,4-Dihydroxyphenylalanine) Cat. No.: HY-N0304

L-DOPA is a natural form of DOPA used in thetreatment of Parkinson's disease. L-DOPA is theprecursor of dopamine and product of tyrosinehydroxylase.

Purity: 99.83%Clinical Data: LaunchedSize: 200 mg, 1 g

L-Hyoscyamine (Daturine) Cat. No.: HY-N0471

L-Hyoscyamine is a chemical compound, a tropanealkaloid it is the levo-isomer to atropine.


L-Praziquanamine ((+)-Praziquanamine) Cat. No.: HY-N1765

L-Praziquanamine is a natural product.


L-Stepholidine (Stepholidine; (-)-Stepholidine; L-SPD) Cat. No.: HY-N6960

L-Stepholidine (Stepholidine), an alkaloid extractof the Chinese herb , is theStephania intermediafirst compound known to exhibit mixed dopamine

agonist/D2 antagonist properties.D1 receptor


Lappaconitine ((+)-Lappaconitine) Cat. No.: HY-N0383

Lappaconitine, isolated from Aconitum sinomontanumNakai, was characterized as analgesic principle.IC50 value: Target: In vitro: In vivo:Lappaconitine was characterized as analgesicprinciple by our laboratory.


Lappaconitine hydrobromide (Allapinine) Cat. No.: HY-N0118

Lappaconitine hydrobromide, a diterpene alkaloid,is a drug for the treatment of cardiacarrhythmias.


Latrunculin A (LAT-A) Cat. No.: HY-16929

Latrunculin A (LAT-A) is a toxin isolated from thered sea sponge , binds toLatrunculia magnificaactin monomers, inhibits polymerization of actin,with s of 0.1, 0.4, 4.7 μM and 0.19 μM forKd

ATP-actin, ADP-Pi-actin, ADP-actin and G-actin,respectively.

Purity: >95.0%Clinical Data: No Development ReportedSize: 100 μg


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Laurolitsine hydrochloride ((+)-Norboldine hydrochloride) Cat. No.: HY-N2352A

Laurolitsine hydrochloride is an alkaloid isolatedfrom , and shows weakPhoebe formosanaanti-inflammatory activity.


Leonurine (SCM-198) Cat. No.: HY-N0741

Leonurine is an alkaloid isolated from Herba, with anti-oxidative and anti-inflammatory.leonuri


Leonurine hydrochloride (SCM-198 hydrochloride) Cat. No.: HY-N0741A

Leonurine hydrochloride is an alkaloid isolatedfrom , with anti-oxidative andHerba leonurianti-inflammatory.


Levoleucovorin Calcium (Calcium levofolinate; CL307782) Cat. No.: HY-13667

Levoleucovorin calcium is the calcium salt ofLevoleucovorin, which is the enantiomericallyactive form of folinic acid.

Purity: 95.24%Clinical Data: LaunchedSize: 10 mM × 1 mL, 100 mg, 500 mg, 1 g, 2 g

Ligustrazine hydrochloride (Chuanxiongzine hydrochloride;

Tetramethylpyrazine hydrochloride) Cat. No.: HY-N0935

Ligustrazine (hydrochloride) is a natural product.IC50 value: Target: In vitro: Ligustrazinehydrochloride displayed a protection effect oninjured ECV304 cells, NOS and NO formation weresignificantly increased compared with the modelgroup . In vivo:.


Lisinopril (MK-521) Cat. No.: HY-18206

Lisinopril (MK-521) is angiotensin-convertingenzyme inhibitor, used in treatment ofhypertension, congestive heart failure, and heartattacks.


Lobeline hydrochloride (α-Lobeline hydrochloride; L-Lobeline hydrochloride) Cat. No.: HY-B0979

Lobeline hydrochloride, a nicotinic receptoragonist, acting as a potent antagonist at bothα3β2 and α4β2 neuronal nicotinic receptorsubtypes.


LudaconitineCat. No.: HY-N6816

Ludaconitine, isolated from Aconitum (Bruhl) Stapf, exhibitsspicatum

antileishmanial activity with an IC of 36.1050

μg/mL.


Lycorine hydrochlorideCat. No.: HY-N0289

Lycorine (hydrochloride) is VE-cadherininhibitor,and has IC50 of 1.2μM in Hey1B cell.


LysergolCat. No.: HY-N6809

Lysergol, a clavine alkaloid isolated from seedsof , is a bioenhancer forIpomoea muricatathe drugs and nutrients and has antibacterialactivity. Lysergol has been used as hypotensive,psychotropic analgesic and uterus- andintestine-stimulating drug.



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Matrine (Matridin-15-one; Vegard; α-Matrine) Cat. No.: HY-N0164

Matrine (Matridin-15-one) is an alkaloid found inplants from the Sophora genus. It has a variety ofpharmacological effects, including anti-cancereffects, and action as a kappa opioid receptor andu-receptor agonist.


MedetomidineCat. No.: HY-17034

Medetomidine(Domtor) is a potent, highly selectiveα2-adrenoceptor agonist (Ki values are 1.08 and1750 nM for α2- and α1-adrenoceptorsrespectively).

Purity: 99.88%Clinical Data: LaunchedSize: 5 mg, 10 mg, 50 mg

MeleagrinCat. No.: HY-N6797

Meleagrin is a roquefortine C-derived alkaloidproduced by fungi of the genus andPenicilliumhas antimicrobial and anti-proliferativeactivities. Meleagrin is a class of inhibitor.FabI


Meropenem (SM 7338) Cat. No.: HY-13678

Meropenem (SM 7338) is a carbapenem antibiotic,which displaying a broad spectrum of antibacterialactivity.


MesaconineCat. No.: HY-N1922

Mesaconinean, an ingredient from Aconitum Debx., has cardiac effect.carmichaelii


MesaconitineCat. No.: HY-N0724

Mesaconitine is the main active component of genusaconitum plants.


Mianserin hydrochloride (Org GB 94) Cat. No.: HY-B0188A

Mianserin hydrochloride is a H1 receptor inverseagonist and is a psychoactive agent of thetetracyclic antidepressant. Target: H1 receptorMianserin is a psychoactive drug of thetetracyclic antidepressant (TeCA) therapeuticfamily.


Monocrotaline N-OxideCat. No.: HY-N6828

Monocrotaline N-Oxide, a monocrotaline metabolite,leads to DNA adduct formation in vivo.


MoxifloxacinCat. No.: HY-66011A

Moxifloxacin is a synthetic fluoroquinoloneantibiotic agent.


N-Benzylpalmitamide (N-Benzylhexadecanamide; Macamide 1) Cat. No.: HY-N2365

N-Benzylpalmitamide is a macamide isolated from, acts as an inhibitor ofLepidium meyenii

.fatty acid amide hydrolase (FAAH)



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N-Methylcytisine (Caulophylline) Cat. No.: HY-N0443

N-Methylcytisine (Caulophylline), a tricyclicquinolizidine alkaloid, exerts hypoglycaemic,analgesic and anti-inflammatory activities.


N-NornuciferineCat. No.: HY-N2129

N-Nornuciferine is an aporphine alkaloid in lotusleaf that significantly inhibits with CYP2D6 IC50

and of 3.76 and 2.34 μM, respectively.Ki


N-trans-Feruloyltyramine (N-feruloyltyramine; Moupinamide) Cat. No.: HY-N2410

N-trans-Feruloyltyramine (N-feruloyltyramine), analkaloid from , is an inhibitor of Piper nigru COX1and , with potential antioxidant properties.COX2N-trans-Feruloyltyramine possessesanti-inflammatory activity.


N-BenzyllinolenamideCat. No.: HY-N3033

N-Benzyllinolenamide is a natural macamideisolated from , acts as anLepidium meyeniiinhibitor of fatty acid amide hydrolase ( )FAAHwith an of 41.8 μM.IC50


N6-Methyladenosine (6-Methyladenosine; N-Methyladenosine) Cat. No.: HY-N0086

N6-Methyladenosine is the most prevalent internal(non-cap) modification present in the messengerRNA (mRNA) of all higher eukaryotes.


Narciclasine (Lycoricidinol) Cat. No.: HY-16563

Narciclasine is a plant growth modulator.Narciclasine modulates the Rho/Rho kinase/LIMkinase/cofilin signaling pathway, greatlyincreasing GTPase RhoA activity as well asinducing actin stress fiber formation in aRhoA-dependent manner.


Neferine ((-)-Neferine) Cat. No.: HY-N0441

Neferine is a major bisbenzylisoquinline alkaloid.Neferine strongly inhibits activation.NF-κB


NeotuberostemonineCat. No.: HY-N3196

Neotuberostemonine, one of the main antitussivealkaloids in the root of Stemona tuberosa Lour,attenuates bleomycin-induced pulmonary fibrosis bysuppressing the recruitment and activation ofmacrophages.


NicergolineCat. No.: HY-B0702

Nicergoline is an ergot derivative used to treatsenile dementia and other disorders with vascularorigins. Target: Alpha-1A adrenergic receptorNicergoline acts by inhibiting the postsynapticalpha(1)-adrenoceptors on vascular smooth muscle.


Nifuratel (NF 113; SAP 113; Methylmercadone) Cat. No.: HY-A0059

Nifuratel(NF 113, SAP 113) is a broadantibacterial spectrum agent, which is used as anantibacterial, antifungal, and antiprotozoal(Trichomonas).



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NigakinoneCat. No.: HY-N2128

Nigakinone is one of the most abundant alkaloidsresponsible for the major pharmacologicalactivities of Kumu.


Nonivamide (Pseudocapsaicin; Pelargonic acid vanillylamide;

Nonanoic acid vanillylamide) Cat. No.: HY-17568

Nonivamide is a <b<TRPV1 agonist, whichexhibits 4d- value of 5.1 mg/L in staticEC50

toxicity tests.

Purity: 98.15%Clinical Data: LaunchedSize: 10 mM × 1 mL, 100 mg, 500 mg, 5 g

Norfloxacin hydrochloride (MK-0366 (hydrochloride)) Cat. No.: HY-B0132A

Norfloxacin (hydrochloride) (MK-0366(hydrochloride)) is a broad-spectrum antibioticthat is active against both Gram-positive andGram-negative bacteria, which functions byinhibiting DNA gyrase.


Norisoboldine ((+)-Laurelliptine) Cat. No.: HY-N0586

Norisoboldine is an isoquinoline alkaloid whichacts as an AhR agonist, and enhances the functionof the .adenosine A1 receptor


NuciferineCat. No.: HY-N0049

Nuciferine is an antagonist at ( =4785-HT2A IC50

nM), ( =131 nM), and ( =15-HT2C IC50 5-HT2B IC50

μM), an inverse agonist at ( =150 nM),5-HT7 IC50

a partial agonist at ( =64 nM), D2 EC50 D5

( =2.6 μM) and ( =700 nM), anEC50 5-HT6 EC50

agonist at ( =3.2 μM) and…5-HT1A EC50


Orotic acid (6-Carboxyuracil; Vitamin B13) Cat. No.: HY-N0157

Orotic acid (OA) is an intermediate in pyrimidinemetabolism.


Oxaceprol (N-Acetyl-L-hydroxyproline) Cat. No.: HY-17490

Oxaceprol is an anti-inflammatory drug used in thetreatment of osteoarthritis.

Purity: >95.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 1 g

Oxcarbazepine (GP 47680) Cat. No.: HY-B0114

Oxcarbazepine (GP 47680) inhibits the binding of[3H]BTX to sodium channels with IC of 160 μM and50

also inhibits the influx of 22Na+ into rat brainsynaptosomes with IC about 100 μM.50


Oxindole (Indolin-2-one) Cat. No.: HY-Y0061

Oxindole (Indolin-2-one) is an aromaticheterocyclic building block. 2-indolinonederivatives have become lead compounds in theresearch of kinase inhibitors.


Oxyberberin (Berlambine; 8-Oxoberberine; Ketoberberine) Cat. No.: HY-N5027

Berlambine is a natural alkaloid isolated frommany plants.



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https://www.MedChemExpress.com/Orotic-acid.html

https://www.MedChemExpress.com/Oxaceprol.html

https://www.MedChemExpress.com/Oxcarbazepine.html

https://www.MedChemExpress.com/NSC_274863.html

https://www.MedChemExpress.com/oxyberberin.html

OxymatrineCat. No.: HY-N0158

Oxymatrine, an alkaloid from the roots of Sophoraspecies, with anti-inflammatory, antifibrosis, andantitumor effects, inhibits the expression andiNOS

pathway.TGF-β/Smad

Purity: >98.0%Clinical Data: Phase 4Size: 10 mM × 1 mL, 100 mg, 200 mg, 500 mg, 1 g

p-SynephrineCat. No.: HY-113236

p-Synephrine is an organic compound, found inmultiple biofluids, such as urine and blood.


Palmatine chlorideCat. No.: HY-N0110

Palmatine chloride an isoquinoline alkaloid, is animportant medicinal herbal extract with diversepharmacological and biological properties.

Purity: 95.97%Clinical Data: No Development ReportedSize: 10 mM × 1 mL, 250 mg, 1 g

ParaxanthineCat. No.: HY-W016498

Paraxanthine, a caffeine metabolite, providesprotection against Dopaminergic cell death viastimulation of Ryanodine Receptor Channels.


PaxillineCat. No.: HY-N6778

Paxilline is an indole alkaloid mycotoxin from, acts as a potent BKPenicillium paxilli

channels inhibitor by an almost exclusivelyclosed-channel block mechanism.


Pefloxacin (Pefloxacinium) Cat. No.: HY-B0147

Pefloxacin is a an antibacterial agent andprevents bacterial DNA replication by inhibitingDNA gyrase (topoisomerse) Target: DNA gyrasePefloxacin is a synthetic chemotherapeutic agentused to treat severe and life-threateningbacterial infections.


Peimine (Verticine; Dihydroisoimperialine) Cat. No.: HY-N0212

Peimine(Dihydroisoimperialine; Verticine) is anatural compound with good anti-inflammatoryeffects in vivo.


Peiminine (Verticinone; Raddeanine) Cat. No.: HY-N0213

Peiminine(Verticinone; Raddeanine) is a naturalcompound with anti-inflammatory activity. IC50value: Target: Peiminine and DXS significantlyreduced alveolar inflammation and pulmonaryinterstitial inflammation in rats withbleomycin-induced lung injury.


Peimisine (Ebeiensine) Cat. No.: HY-N0214

Peimisine(Ebeiensine) is a steroidal alkaloidwhich is the major biologically active componentin Bulbus Fritillariae; possess a variety oftoxicological and pharmacological effects onhumans.


Pemetrexed (LY231514) Cat. No.: HY-10820

Pemetrexed is a novel , the values ofantifolate Ki

the pentaglutamate of LY231514 are 1.3, 7.2, and65 nM for inhibits thymidylate synthase ( ),TSdihydrofolate reductase ( ), and glycinamideDHFRribonucleotide formyltransferase ( ),GARFTrespectively.



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https://www.MedChemExpress.com/Palmatine-chloride.html

https://www.MedChemExpress.com/Paraxanthine.html

https://www.MedChemExpress.com/paxilline.html

https://www.MedChemExpress.com/pefloxacin.html

https://www.MedChemExpress.com/Peimine.html

https://www.MedChemExpress.com/Peiminine.html

https://www.MedChemExpress.com/Peimisine.html

https://www.MedChemExpress.com/pemetrexed.html

Pemetrexed disodium (LY231514 disodium) Cat. No.: HY-10820A

Pemetrexed disodium is a novel thatantifolateinhibits the folatedependent enzymes

, ,thymidylate synthase dihydrofolate reductaseand glycinamide ribonucleotide

with s of 1.3, 7.2, and 65formyltransferase Ki

nM, respectively.


Penitrem ACat. No.: HY-N6776

Penitrem A is an indole diterpene neurotoxicalkaloid produced by , acts as aPenicilliumselective antagonist withBK channelantiproliferative and anti-invasive activitiesagainst multiple malignancies.


Perindopril (S-9490) Cat. No.: HY-B0130

Perindopril is a long-acting ACE inhibitor ofwhich is used to treat high blood pressure, heartfailure or stable coronary artery disease. Target:ACE Perindopril is a long-acting ACE inhibitor.


Pilocarpine HydrochlorideCat. No.: HY-B0726

Pilocarpine Hydrochloride is a selective M3-typemuscarinic acetylcholine receptor (M3

) agonist.muscarinic receptor

Purity: 99.92%Clinical Data: LaunchedSize: 100 mg, 500 mg

Pioglitazone (U 72107) Cat. No.: HY-13956

Pioglitazone is a potent and selective PPARγagonist with high affinity binding to the PPARγligand-binding domain with of 0.93 and 0.99EC50

μM for human and mouse PPARγ, respectively.


Piperine (Bioperine; 1-Piperoylpiperidine) Cat. No.: HY-N0144

Piperine, a natural alkaloid isolated from Piper L, inhibits and nigrum P-glycoprotein CYP3A4

activities with an value of 61.94±0.054 μg/mLIC50

in HeLa cell.

Purity: 98.76%Clinical Data: Phase 2Size: 10 mM × 1 mL, 200 mg, 1 g, 5 g

Piperlongumine (Piplartine) Cat. No.: HY-N2329

Piperlongumine is a natural alkaloid isolated from Linn, possesses ant-inflammatory,Piper longum

antibacterial, antiangiogenic, antioxidant,antitumor, and antidiabetic activities.Piperlongumine induces ROS, and induces apoptosisin cancer cell lines.


Piperlotine CCat. No.: HY-N3049

Piperlotine C is an alkaloid isolated from Piper, with anti-platelet aggregation induced bylolot

arachidonic acid, and the is 26.6 µg/mL.IC50


Pirmenol hydrochloride (Cl-845; (±)-Pirmenol hydrochlorid) Cat. No.: HY-100795A

Pirmenol hydrochloride inhibits by blockingIK.ACh

. The of Pirmenol formuscarinic receptors IC50

inhibition of Carbachol-induced I is 0.1 μM.K.ACh

Purity: 95.63%Clinical Data: LaunchedSize: 10 mM × 1 mL, 1 mg, 5 mg, 10 mg, 50 mg, 100 mg

Pizotifen malate (BC-105 (malate); Pizotyline (malate)) Cat. No.: HY-B0115A

Pizotifen (malate) (BC-105 (malate)) is a potent receptor antagonist, with a high affinity5-HT2

for binding site.5-HT1C



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https://www.MedChemExpress.com/Piperine.html

https://www.MedChemExpress.com/Piperlongumine.html

https://www.MedChemExpress.com/piperlotine-c.html

https://www.MedChemExpress.com/Pirmenol-hydrochloride.html

https://www.MedChemExpress.com/pizotifen-malate.html

PrazosinCat. No.: HY-B0193

Prazosin is an alpha-adrenergic blocker and is asympatholytic drug used to treat high bloodpressure and anxiety, PTSD, and panic disorder.Target: Adrenergic Receptor Prazosin, is asympatholytic drug used to treat high bloodpressure and anxiety, PTSD, andpanic disorder.


Protopine (Corydinine) Cat. No.: HY-N0793

Protopine, an isoquinoline alkaloid contained inplants in northeast Asia.


QuinidineCat. No.: HY-B1751

Quinidine is an antiarrhythmic agent for thetreatment of abnormal heart rhythms and alsomalaria.


Rauwolscine hydrochloride (α-Yohimbine hydrochloride;

Corynanthidine hydrochloride; Isoyohimbine hydrochloride) Cat. No.: HY-12710A

Rauwolscine hydrochloride is a potent and specific receptor antagonist with a of 12α2 adrenergic Ki

nM.


ReserpineCat. No.: HY-N0480

Reserpine is an inhibitor of the vesicular ( ).monoamine transporter 2 VMAT2


Reserpine hydrochlorideCat. No.: HY-N0480A

Reserpine hydrochloride is an inhibitor of the ( ).vesicular monoamine transporter 2 VMAT2


RhynchophyllineCat. No.: HY-N0387

Rhyncholphylline, an alkaloid isolated fromUncaria, shows potent inhibition oflipopolysaccharide (LPS)-induced NO production inrat primary microglial cells.


Roquinimex (Linomide; FCF89; ABR212616) Cat. No.: HY-13743

Roquinimex (Linomide; PNU212616; ABR212616) is aquinoline derivative immunostimulant whichincreases NK cell activity and macrophagecytotoxicity; inhibits angiogenesis and reducesthe secretion of TNF alpha.


Rotundine ((-)-Tetrahydropalmatine; L-Tetrahydropalmatine) Cat. No.: HY-N0096

Rotundine is an antagonist of , dopamine D1 D2and with s of 166 nM, 1.4 μMD3 receptors IC50

and 3.3 μM, respectively. Rotundine is also anantagonist of with an of 370 nM.5-HT1A IC50


Rubitecan (RFS 2000; 9-Nitrocamptothecin) Cat. No.: HY-13744

Rubitecan (RFS 2000), a Camptothecin derivative,is an orally active inhibitortopoisomerase Iwith broad antitumor activity, and inducesprotein-linked DNA single-strand breaks, therebyblocking DNA and RNA synthesis in dividing cells.



https://www.MedChemExpress.com/Prazosin.html

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https://www.MedChemExpress.com/Quinidine.html

https://www.MedChemExpress.com/Rauwolscine_hydrochloride.html

https://www.MedChemExpress.com/Reserpine.html

https://www.MedChemExpress.com/reserpine-hydrochloride.html

https://www.MedChemExpress.com/Rhynchophylline.html

https://www.MedChemExpress.com/Roquinimex.html

https://www.MedChemExpress.com/Rotundine.html

https://www.MedChemExpress.com/rubitecan.html

Rufinamide (CGP 33101; E 2080; RUF 331) Cat. No.: HY-A0042

Rufinamide(E 2080; CGP 33101; RUF 331) is a newantiepileptic agent that differs structurally fromother antiepileptic drugs and is approved asadjunctive therapy for Lennox-Gastaut syndrome(LGS).


Rutaecarpine (Rutecarpine) Cat. No.: HY-N0147

Rutaecarpine, an alkaloid of , isEvodia rutaecarpaan inhibitor of with an value of 0.28COX-2 IC50

μM.


Salsolidine (6,7-Dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline) Cat. No.: HY-22385

Salsolidine is a tetrahydroisoquinoline alkaloid,acts as a stereoselective competitive MAO Ainhibitor.


Sanguinarine (Pseudochelerythrine; Sanguinarin) Cat. No.: HY-N0052

Sanguinarine, a benzophenanthridine alkaloidderived from the root of , canSanguinaria Canadensisstimulate via activating the productionapoptosisof reactive oxygen species (ROS).Sanguinarine-induced apoptosis is associated withthe activation of JNK and NF-κB.


Sanguinarine chloride (Pseudochelerythrine chloride; Sanguinarium chloride) Cat. No.: HY-N0052A

Sanguinarine chloride, a benzophenanthridinealkaloid derived from the root of Sanguinaria

, can stimulate via activatingCanadensis apoptosisthe production of reactive oxygen species (ROS).Sanguinarine-induced apoptosis is associated withthe activation of JNK and NF-κB.


Santacruzamate A (CAY-10683) Cat. No.: HY-N0931

Santacruzamate A (CAY-10683) is a potent andselective inhibitor with an of 119 pM.HDAC2 IC50


Sapropterin dihydrochloride (6R-BH4 dihydrochloride;

6R-Tetrahydro-L-biopterin dihydrochloride) Cat. No.: HY-A0124A

Sapropterin dihydrochloride is a synthetic form ofBH4 that is approved for the treatment of BH4responsive PKU.


Sauristolactam (Saurolactam) Cat. No.: HY-118482

Sauristolactam, a natural aristolactam isolatedfrom aerial portions of , hasSaururus chinensissignificant neuroprotective activity againstglutamate-induced toxicity in primary cultured ratcortical cells.


SchinifolineCat. No.: HY-N4164

Schinifoline, a 4-quinolinone derivative isolatedfrom Sieb, improvesZanthoxylum schinifoliumradiosensitizing effect, and effects cell cycleand apoptotic-inducing effects in cancer .


Scopine (6,7-Epoxytropine) Cat. No.: HY-B0459

Scopine is the metabolite of anisodine, which is aα1-adrenergic receptor agonist and used in thetreatment of acute circulatory shock.



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https://www.MedChemExpress.com/Sanguinarine.html

https://www.MedChemExpress.com/Sanguinarine-chloride.html

https://www.MedChemExpress.com/Santacruzamate-A.html

https://www.MedChemExpress.com/Sapropterin-dihydrochloride.html

https://www.MedChemExpress.com/Sauristolactam.html

https://www.MedChemExpress.com/schinifoline.html

https://www.MedChemExpress.com/scopine.html

Scopolamine (Hyoscine; Scopine (-)-tropate; Scopine tropate) Cat. No.: HY-N0296

Scopolamine is a high affinity (nM) muscarinicantagonist. receptor-responses are5-HT3

reversibly inhibited by Scopolamine with an IC50

of 2.09 μM.


Scopolamine butylbromide (Hyoscine butylbromide;

(-)-Scopolamine butylbromide; Butylscopolamine bromide) Cat. No.: HY-N0340

Scopolamine butylbromide is a competitiveantagonist of muscarinic acetylcholine receptor(mAChR) with an IC50 of 55.3 ± 4.3 nM.


Scopolamine hydrobromide ((-)-Scopolamine hydrobromide;

Hyoscine hydrobromide; Scopine hydrobromide) Cat. No.: HY-N0296A

Scopolamine hydrobromide is a high affinity (nM) antagonist. muscarinic 5-HT3

receptor-responses are reversibly inhibited byScopolamine with an of 2.09 μM.IC50


Senecionine (Senecionan-11,16-dione, 12-hydroxy-; Aureine; Senecionin) Cat. No.: HY-N2560

Senecionine is a pyrrolizidine alkaloid isolatedfrom . Senecionine is toxic toSenecio vulgarisanimals and humans.


SeneciphyllinineCat. No.: HY-N1283

Seneciphyllinine, a pyrrolizidine alkaloid, isisolated from the roots of .Gynura japonicaPyrrolizidine alkaloids are highly hepatotoxicnatural chemicals that produce irreversiblechronic and acute hepatotoxic effects on humanbeings.


Setiptiline maleate (MO-8282) Cat. No.: HY-32329A

Setiptiline is a serotonin receptor antagonist.


SinapineCat. No.: HY-N5077

Sinapine is an alkaloid from seeds of thecruciferous species which shows favorablebiological activities such as antioxidant andradio-protective activities.


Sinapine thiocyanateCat. No.: HY-N0450

Sinapine thiocyanate is an alkaloid from seeds ofthe cruciferous species which shows favorablebiological activities such as antioxidant andradio-protective activities.


Sinomenine hydrochloride (Cucoline hydrochloride) Cat. No.: HY-15122A

Sinomenine hydrochloride is a blocker of the activation and also an activator of NF-κB μ-opioid

.receptor


Sipeimine (Imperialine) Cat. No.: HY-N0696

Sipeimine is a natural product isolated fromFritillaria ussuriensis.



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https://www.MedChemExpress.com/Senecionine.html

https://www.MedChemExpress.com/seneciphyllinine.html

https://www.MedChemExpress.com/setiptiline-maleate.html

https://www.MedChemExpress.com/Sinapine.html

https://www.MedChemExpress.com/Sinapine-thiocyanate.html

https://www.MedChemExpress.com/Sinomenine_hydrochloride.html

https://www.MedChemExpress.com/Sipeimine.html

Solamargine (Solamargin; δ-Solanigrine) Cat. No.: HY-N0069

Solamargine is a major steroidal alkaloidglycoside extracted from a traditional Chinesemedicinal herb, Solanum nigrum L. (SNL); has beenshown to inhibit growth and induce apoptosis ofvarious cancer cells.


Solasodine (Purapuridine; Solancarpidine; Solasodin) Cat. No.: HY-N0068

Solasodine(Purapuridine) is a poisonous alkaloidchemical compound that occurs in plants of theSolanaceae family. Solasodine showed selectivecytotoxicity against cervical cancer cell line(HeLa) and human myeloid leukemia cell line(U937).


SophocarpineCat. No.: HY-N0103

Sophocarpine is one of the significant alkaloidextracted from the traditional herb medicine

which has many pharmacologicalSophora flavescensproperties such as anti-virus, anti-tumor,anti-inflammatory.


Sophocarpine (monohydrate)Cat. No.: HY-N0103A

Sophocarpine (monohydrate) is one of thesignificant alkaloid extracted from thetraditional herb medicine whichSophora flavescenshas many pharmacological properties such asanti-virus, anti-tumor, anti-inflammatory.


Stachydrine hydrochlorideCat. No.: HY-N0738

Stachydrine hydrochloride is the major activeconstituent of , which is a potentialHerba Leonuritherapy for cardiovascular diseases. Stachydrinecan inhibit the signal pathway.NF-κBAnti-hypertrophic activities.


Staurosporine (Antibiotic AM-2282; STS; AM-2282) Cat. No.: HY-15141

Staurosporine is a potent and non-selectiveinhibitor of protein kinases with s of 6 nM,IC50

15 nM, 2 nM, and 3 nM for , , , andPKC PKA c-Fgr respectively.Phosphorylase kinase


SulfapyridineCat. No.: HY-B0212

Sulfapyridine(Dagenan) is a sulfonamideantibacterial.

Purity: 99.96%Clinical Data: LaunchedSize: 1 g, 5 g

SulfathiazoleCat. No.: HY-B0507

Sulfathiazole is an organosulfur compound that hasbeen used as a short-acting sulfa drug. Target:Antibacterial Sulfathiazole (20 μg/L) starts to bedegraded between day 31 and day 38 in one of thetwo batch reactors containing different wastewatermatrices.

Purity: >98%Clinical Data: LaunchedSize: 1 g

Swainsonine (Tridolgosir) Cat. No.: HY-N6722

Swainsonine is an alkaloid isolated from, acts as an inhibitor ofAstragalus

, with anti-tumor activity.α-mannosidase


Synephrine hydrochloride (Oxedrine hydrochloride) Cat. No.: HY-N0132A

Synephrine hydrochloride (Oxedrine hydrochloride)is an alkaloid. Synephrine hydrochloride (Oxedrinehydrochloride) produces most of its biologicaleffects by acting as an agonist at adrenergicreceptors.



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https://www.MedChemExpress.com/Stachydrine_hydrochloride.html

https://www.MedChemExpress.com/Staurosporine.html

https://www.MedChemExpress.com/sulfapyridine.html

https://www.MedChemExpress.com/sulfathiazole.html

https://www.MedChemExpress.com/swainsonine.html

https://www.MedChemExpress.com/synephrine-hydrochloride.html

Talipexole (B-HT 920) Cat. No.: HY-A0040

Talipexole (B-HT920) is a dopamine agonist thathas been proposed as an antiparkinsonian agent.Target: Dopamine Receptor B-HT920 is a selectivealpha 2-adrenoceptor agonist.


Tandospirone citrate (SM-3997 citrate) Cat. No.: HY-B0061

Tandospirone citrate is a potent and selective5-HT1A receptor partial agonist (Ki = 27 nM) thatdisplays selectivity over SR-2, SR-1C, α1, α2, D1and D2 receptors (Ki values ranging from1300-41000 nM).


TerazosinCat. No.: HY-B0371

Terazosin is a selective alpha1-antagonist usedfor treatment of symptoms of benign prostatichyperplasia (BPH).


Tetrahydroberberine (Canadine) Cat. No.: HY-N0925

Tetrahydroberberine is an isoquinoline alkaloidisolated from corydalis tuber; has micromolaraffinity for dopamine D(2) (pK(i) = 6.08) and5-HT(1A) (pK(i) = 5.38) receptors but moderate tono affinity for other relevant serotonin receptors(5-HT(1B), 5-HT(1D), 5-HT(3), and 5-HT(4);…


Tetrahydrocoptisine ((RS)-Stylopine; (±)-Stylopin) Cat. No.: HY-N0924

Tetrahydrocoptisine is an alkaloid compoundoriginally isolated from Corydalis tubers thatexhibits anti-inflammatory and anti-parasiticactivities.


Tetrahydropalmatine (DL-Tetrahydropalmatine) Cat. No.: HY-N0300

Tetrahydropalmatine, an active component isolatedfrom corydalis, acts through inhibition ofamygdaloid release of to inhibit andopamineepileptic attack in rats.


Tetramethylpyrazine (Ligustrazine) Cat. No.: HY-N0264

Tetramethylpyrazine (Ligustrazine), analkylpyrazine isolated from Ligusticum

( ), is present in frenchwallichii Chuan Xiongfries, bread, cooked meats, tea, cocoa, coffee,beer, spirits, peanuts, filberts, dairy productsand soy products as fragrance and…


Theobromine (3,7-Dimethylxanthine) Cat. No.: HY-N0138

Theobromine is a methylxanthine found in cacaobeans which can inhibit adenosine receptor A1( ) signaling.AR1

Purity: 99.65%Clinical Data: Phase 3Size: 10 mM × 1 mL, 100 mg

Theophylline (1,3-Dimethylxanthine; Theo-24) Cat. No.: HY-B0809

Theophylline is a nonselective phosphodiesterase inhibitor, blocker, and(PDE) adenosine receptor

activator.histone deacetylase (HDAC)

Purity: 99.94%Clinical Data: LaunchedSize: 10 mM × 1 mL, 5 g

Thymidine (DThyd; Deoxyribothymidine; Deoxythymidine; NSC

21548; Thymidin) Cat. No.: HY-N1150

Thymidine is a a pyrimidine deoxynucleoside.



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https://www.MedChemExpress.com/terazosin.html

https://www.MedChemExpress.com/Tetrahydroberberine.html

https://www.MedChemExpress.com/Tetrahydrocoptisine.html

https://www.MedChemExpress.com/Tetrahydropalmatine.html

https://www.MedChemExpress.com/Tetramethylpyrazine.html

https://www.MedChemExpress.com/Theobromine.html

https://www.MedChemExpress.com/Theophylline.html

https://www.MedChemExpress.com/Thymidine.html

ThymineCat. No.: HY-W010450

Thymine is one of the four nucleobases in thenucleic acid of DNA and can be a target foractions of 5-fluorouracil (5-FU) in cancertreatment, with a K of 2.3 μM.m


Tiagabine (NO050328; NO328; TGB) Cat. No.: HY-B0696

Tiagabine (NO050328) is a potent and selective inhibitor, used as anGABA reuptake

anticonvulsant agent, with s of 67, 446 andIC50

182 nM for [ H]GABA uptake in Synaptosomes,3

Neurons and Glia, respectively.


Tigecycline (GAR-936) Cat. No.: HY-B0117

Tigecycline (GAR-936) is a broad-spectrumglycylcycline antibiotic. The mean inhibitoryconcentration (MIC) of Tigecycline for E. coli(MG1655 strain) is approximately 125 ng/mL.


TomatidineCat. No.: HY-N2149

Tomatidine acts as an anti-inflammatory agent byblocking and signaling.NF-κB JNK

Purity: >98.0%Clinical Data: No Development ReportedSize: 25 mg, 50 mg, 100 mg

Tomatine (α-Tomatine; Lycopersicin; Tomatin) Cat. No.: HY-N2166

Tomatine is a glycoalkaloid, found in the tomatoplant ( Mill.). TomatineLycopersicon esculentumelicits neurotoxicity in RIP1 kinase andcaspase-independent manner. Tomatine promotes theupregulation of nuclear apoptosis inducing factor(AIF) in neuroblastoma cells.


Trabectedin (Ecteinascidin 743; ET-743) Cat. No.: HY-50936

Trabectedin (Ecteinascidin-743 or ET-743) is anovel antitumour agent of marine origin withpotent antitumour activity both in vitro and invivo.

Purity: 99.83%Clinical Data: LaunchedSize: 1 mg

Trigonelline (Trigenolline) Cat. No.: HY-N0414

Trigonelline, an alkaloid with potentialantidiabetic activity, is present in considerableamounts in coffee.


Trigonelline chloride (Trigonelline hydrochloride) Cat. No.: HY-N0415

Trigonelline chloride, an alkaloid with potentialantidiabetic activity, is present in considerableamounts in coffee.


Tropisetron (SDZ-ICS-930 (free base)) Cat. No.: HY-B0072

Tropisetron (SDZ-ICS-930 free base) is a selective5-HT3 receptor antagonist and α7-nicotinicreceptor agonist with an IC50 of 70.1 ± 0.9 nM for5-HT3 receptor.

Purity: >98.0%Clinical Data: LaunchedSize: 10 mM × 1 mL, 10 mg, 50 mg, 100 mg

TryptamineCat. No.: HY-B2132

Tryptamine is a monoamine alkaloid, similar toother trace amines, is believed to play a role asa neuromodulator or neurotransmitter.



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https://www.MedChemExpress.com/Trigonelline_chloride.html

https://www.MedChemExpress.com/tropisetron.html

https://www.MedChemExpress.com/Tryptamine.html

Veratramine (NSC17821; NSC23880) Cat. No.: HY-N0837

Veratramine(NSC17821; NSC23880) is useful as asignal transduction inhibitor for treating tumors.


VicineCat. No.: HY-N2093

Vicine, an alkaloid glycoside found mainly in favabeans, is toxic in individuals and may causehaemolytic anaemia.


Vinblastine sulfate (Vincaleukoblastine sulfate salt) Cat. No.: HY-13780

Vinblastine sulfate is a cytotoxic alkaloid usedagainst various cancer types. Vinblastine sulfateinhibits the formation of microtubule andsuppresses nAChR with an of 8.9 μM.IC50

Purity: 99.85%Clinical Data: LaunchedSize: 10 mM × 1 mL, 5 mg, 10 mg, 50 mg, 100 mg

VincamineCat. No.: HY-B1021

Vincamine is a peripheral vasodilator, thatincreases blood flow to the brain.


Vincristine sulfate (Leurocristine sulfate; 22-Oxovincaleukoblastine sulfate) Cat. No.: HY-N0488

Vincristine sulfate is an antitumor vinca alkaloidwhich inhibits formation in mitoticmicrotubulespindle, resulting in an arrest of dividing cellsat the metaphase stage. It binds to microtubulewith a of 85 nM.Ki

Purity: 99.66%Clinical Data: LaunchedSize: 10 mg, 50 mg, 100 mg, 200 mg

VinflunineCat. No.: HY-B0628

Vinflunine is a new vinca alkaloid uniquelyfluorinated with the properties ofmitotic-arresting and tubulin-interactingactivity.


WilforineCat. No.: HY-N0899

Wilforine is a sesquiterpene pyridine alkaloid;important bioactive compound in T. wilfordiiplants, and is effective in treating idiopathicpulmonary fibrosis.


Yohimbine HydrochlorideCat. No.: HY-N0127

Yohimbine Hydrochloride is an alpha2-adrenoreceptor antagonist, blocking the pre- andpostsynaptic alpha-2 adrenoreceptors and causingan increased release of noradrenaline anddopamine.

Purity: 99.85%Clinical Data: Phase 4Size: 10 mM × 1 mL, 1 g

Yunaconitine (Guayewuanine B) Cat. No.: HY-N0333

Yunaconitine(Guayewuanine B) is a highly toxicaconitum alkaloid.



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https://www.MedChemExpress.com/Vincamine.html

https://www.MedChemExpress.com/vincristine-sulfate.html

https://www.MedChemExpress.com/vinflunine.html

https://www.MedChemExpress.com/Wilforine.html

https://www.MedChemExpress.com/Yohimbine-Hydrochloride.html

https://www.MedChemExpress.com/Yunaconitine.html

alkaloid - medchemexpress.com · alkaloid alkaloids are a group of naturally occurring chemical...

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