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Page 1: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

2003-2004Nervous System

Pharmacology Review

April 21, 202305:41 PM

Page 2: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Adrenocorticotropin(ACTH)

Anterior pituitary hormoneAnticonvulsant

Stimulates synthesisand release of cortisol

Page 3: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Alfentanil

OpioidGeneral anaesthetic

Intravenous anaesthetic

Page 4: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Amantadine

AntiviralAntiparkinson

Treatment of Influenza A Inhibits replication

at the stage of uncoatingInhibits dopamine release

Page 5: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Amitriptyline

Tricyclic antidepressant (TCA)

Page 6: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Amphetamine

Indirect sympathomimeticDrug of abuse

ADD treatmentStimulant

Page 7: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Atropine

Anticholinergic

AntimuscarinicTreatment for bradycardia,

diarrhea, cholinesterase poisoning

Page 8: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Baclofen

Skeletal muscle relaxantAnxiolytic

GABAB agonist

Page 9: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Benztropine

AnticholinergicAntiparkinson

Muscarinic receptor antagonist

Page 10: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Bethanecol

Cholinomimetic

Muscarinic agonistInduces defecation and

urinationBronchoconstrictor

Page 11: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Bromocriptine

Antiparkinson

Dopamine (D2) agonistInhibits prolactin release

Page 12: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Brupropion

Second generation antidepressant

Page 13: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Buprenorphine

Opioid

Partial agonist

Page 14: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Buspirone

Sedative/hypnoticAnxiolytic

Page 15: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Butorphanol

OpioidAnalgesic

receptor partial agonistor antagonist

Page 16: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Carbamazepine

Anticonvulsant

Page 17: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Carbidopa

Antiparkinson

Peripheral dopa decarboxylase inhibitor

Page 18: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Celecoxib

NSAIDAnti-inflammatory

Cyclooxygenase 2 (COX-2) inhibitor

Page 19: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Chloral hydrate

Sedative/HypnoticGeneral anaesthetic

Acts on GABAA receptor complexSimilar to barbiturates

Page 20: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Chlordiazepoxide

Sedative/hypnoticAnxiolytic

Benodiazepine Acts on GABAA receptor

complex

Page 21: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Chlorpromazine

Antipsychotic

Phenothiazine

Page 22: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Clozapine

Antipsychotic

Page 23: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Cocaine

Indirect sympathomimeticDrug of abuse

Topical anaesthetic

StimulantLocal anaesthetic

Page 24: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Codeine

OpioidAnalgesic

Weak agonist

Page 25: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Dantrolene

Skeletal muscle relaxant

Ryanodine receptor antagonistTreatment for malignant hyperthermia

Page 26: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Deprenyl/selegiline

Antiparkinson

Monoamine oxidase B inhibitor(MAO-I)

Potentiates effects of L-Dopa

Page 27: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Desipramine

Tricyclic antidepressant (TCA)

Page 28: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Dextromethorphan

Opioid

Antitussive

Page 29: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Diazepam

Sedative/hypnoticAnxiolytic

Anticonvulsant

Benzodiazepine Acts on GABAA receptor complex

Page 30: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Diphenoxylate docusate

Antidiarrheal

Opiate

Page 31: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Enflurane

General anaesthetic

Inhaled anaesthetic

Page 32: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Entacapone

Antiparkinson

Peripheral catechol-o-methyltransferase inhibitor

Page 33: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ephedra(Ma Huang)

Dietary supplement

Amphetamine-like stimulant

Page 34: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ethanol

Drug of abuse

Sedative

Page 35: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ethosuximide

Anticonvulsant

Page 36: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Etomidate

General anaesthetic

Intravenous anaesthetic

Page 37: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Fentanyl

OpioidAnalgesic

receptor agonist

Page 38: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Flumazenil

Benzodiazepine antagonist

Acts on GABAA receptor complex

Page 39: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Fluoxetine

Antidepressant

Selective serotonin reuptake inhibitor (SSRI)

Page 40: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Flurazepam

Sedative/Hypnotic

Benzodiazepine Acts on GABAA receptor

complex

Page 41: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ginko biloba

Dietary supplement

Treatment of Alzheimer symptoms

Page 42: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Glutethimide

Sedative/Hypnotic

Page 43: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Haloperidol

Antipsychotic

Page 44: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Halothane

General anaesthetic

Inhaled anaesthetic

Page 45: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Heroin

Drug of abuse

Opioid

Page 46: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Imipramine

Indirect sympathomimeticTricyclic antidepressant (TCA)

Antimicturant

Page 47: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Isoflurane

General anaesthetic

Inhaled anaesthetic

Page 48: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Kava kava

Dietary supplement

Stress relief andtreatment of insomnia

Page 49: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ketamine

General anaestheticDrug of abuse

Sedative

Page 50: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Levodopa

Antiparkinson

Dopamine precursor

Page 51: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Lidocaine

Class I antiarrhythmicLocal anaesthetic

Na+ channel blocker(activated and inactivated channels)

Page 52: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Lithium

Antidepressant

Used to treatmanic/depressive disorder

Page 53: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Loperamide

Antidiarrheal

Opiate

Page 54: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Lorazepam

AnxiolyticAnticonvulsant

BenzodiazepineActs on GABAA receptor complex

Page 55: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Lysergic acid diethylamide

(LSD)

Drug of abuse

Hallucinogen

Page 56: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Marijuana

Drug of abuse

Cannabinoid

Page 57: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Meperidine

Opioid analgesic

receptor agonist

Page 58: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Mepivacaine

Local anaesthetic

Page 59: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Meprobamate

Sedative/hypnoticAnxiolytic

Page 60: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Metamphetamine

Drug of abuse

Stimulant

Page 61: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Methadone

Opioid

receptor agonist

Page 62: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Morphine

OpioidAnalgesic

receptor agonist

Page 63: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nalbuphine

Opioid antagonist

receptor antagonist

Page 64: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nalmefene

Opioid antagonist

Page 65: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nalorphine

Opioid antagonist

Page 66: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Naloxone

Opioid antagonist

Page 67: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Naltrexone

Opioid antagonist

Page 68: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Neostigmine

Anticholinesterase

VasodilatorTreatment for myaesthenia gravisPromotes defecation and urination

Bronchoconstrictor

Page 69: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nicotine

CholinomimeticDrug of abuse

Nicotinic receptor agonist(skeletal muscle contraction)

StimulantSmoking cessation medication

Page 70: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nitrous oxide

General anaesthetic

Inhaled anaesthetic

Page 71: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Nortriptyline

Tricyclic antidepressant (TCA)

Page 72: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Oxazepam

Sedative/hypnoticAnxiolytic

BenzodiazepineActs on GABAA receptor complex

Page 73: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Oxybutinin

Anticholinergic

Muscarinic receptor antagonistPrevents urination

Page 74: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Oxycodone

Analgesic

Opioid agonist

Page 75: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Paraldehyde

Sedative/Hypnotic

Page 76: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Pentazocine

Opioid analgesic

receptor partial agonist or antagonist

Page 77: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Pentobarbital

Sedative/Hypnotic

Barbiturate

Page 78: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Phencyclidine (PCP)

Drug of abuse

Hallucinogen

Page 79: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Phenobarbital

Sedative/HypnoticAnticonvulsant

Barbiturate

Page 80: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Phenytoin

AnticonvulsantClass I antiarrhythmic

Na+ channel blocker(inactivated channels)

Page 81: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Pramipexole

Antiparkinson

Dopamine agonist (non-ergot)

Page 82: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Primidone

Anticonvulsant

Page 83: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Procaine

Local anaesthetic

Page 84: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Propofol

General anaesthetic

Intravenous anaesthetic

Page 85: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Resperidone

Antipsychotic

Page 86: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Ropinirole

Antiparkinson

Dopamine agonist (non-ergot)

Page 87: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Sertraline

Antidepressant

Selective serotonin reuptake inhibitor (SSRI)

Page 88: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Sildenafil

Vasodilator

Promotes erection

Page 89: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

St. John’s Wort

Dietary supplement

Antidepressant

Page 90: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Sufentanil

OpioidGeneral anaesthetic

Intravenous anaesthetic

Page 91: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Temazepam

Sedative/Hypnotic

BenzodiazepineActs on GABAA receptor complex

Page 92: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Tetracaine

Local anaesthetic

Page 93: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Thiopental

General anaesthetic

Ultra-short-acting barbiturate

Page 94: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Thioridazine

Antipsychotic

Phenothiazine

Page 95: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Thiothixene

Antipsychotic

Page 96: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Tolterodine

Anticholinergic

Muscarinic receptor antagonistPrevents urination

Page 97: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Tranylcypromine

Antidepressant

Monoamine oxidase inhibitor (MAO-I)

Page 98: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Triazolam

Sedative/Hypnotic

BenzodiazepineActs on GABAA receptor complex

Page 99: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Trifluoperazine

Antipsychotic

Phenothiazine

Page 100: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Trihexyphenidyl

Antiparkinson

Antimuscarinic

Page 101: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Valproic acid

Anticonvulsant

Page 102: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Vigabatrin

Anticonvulsant

Irreversible GABA aminotransferase inhibitor

Page 103: 2003-2004 Nervous System Pharmacology Review 26 December 2015 9:45 AM

Zolpidem

Sedative/Hypnotic

Non-benzodiazepine