acetyl!choline! cns! norepinephrine gaba - … isoproterenol salmeterol! terbutaline antagonists!...

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Nervous System CNS Brain & spinal cord Acetyl choline Dopamine Serotonin Norepinephrine GABA Glutamate Opioids Somatic Neuromuscular junction Nicotinic (ACh) PNS PSNS Organs, glands Muscarinic (ACh) SNS CV & lung smooth muscle Alpha (NE) Beta (NE) Enteric Many neurotransmitters

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Nervous  System  

CNS   Brain  &  spinal  cord  

Acetyl  choline  

Dopamine  

Serotonin  

Norepinephrine  

GABA  

Glutamate  

Opioids  

Somatic   Neuromuscular  junction   Nicotinic  (ACh)  

PNS  

PSNS   Organs,  glands   Muscarinic  (ACh)  

SNS   CV  &  lung  smooth  muscle  

Alpha  (NE)  

Beta  (NE)  Enteric   Many  

neurotransmitters  

     

PSNS  

Muscarinic  

Bethanechol  

Pilocarpine  

Donepezil  

Neostigmine  

Anti  Muscarinic  

Atropine  

Scopolamine  

1st  Generation  antihistamines  

Tricyclic  antidepressants  

 

CNS  

Acetyl  choline  

Anti-­‐Alzheimer's,  Smoking  cessation,  Antiemetics  

Dopamine  Anti  Parkinson's,  Anti  EPS,  Antipsychotics,  ADHD,  

Antiemetics  

GABA   AEDs,  Sedatives,  Hypnotics,  General  anesthetics  

Glutamate   Ketamine,  Memantine  

Norepinephrine     Antidepressants,  Antipsychotics,  Antihypertensive  

Opioids   Sedation,  Analgesia,  Addiction,  Antitussive,  Antidiarrheal  

Serotonin   Antidepressants,  Antipsychotics,  Antiemetics,  Antimigraine  

 

SNS  

Alpha  

Antagonists  

Alpha  1  

Doxazosin  

Tamsulosin  

Mixed  

Phentolamine  

Agonists  

Alpha  2  

Clonidine  

Mixed  

Ephedrine  

Oxymetazoline  

Phenylephrine  

Pseudoephedrine  

Mixed  Alpha  and  Beta  

Agonists  

Dobutamine  

Catecholamines  

Antagonists  

Labetalol  

Beta  

Agonists  

Albuterol  

Isoproterenol  

Salmeterol  

Terbutaline  

Antagonists  

Atenolol  

Metoprolol  

Propranolol